Search Count: 21
 |
Cryo-Em Structure Of Human Slfn14
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-06-18 Classification: HYDROLASE Ligands: ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-06-18
Ligands: ZN
 |
X-Ray Crystal Structure Of Afssfn From Chaperone Dnajb8.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.75 Å Release Date: 2024-01-31 Classification: CHAPERONE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-31
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-(3-(1-(4-Chlorophenyl)Cyclopropyl) -[1,2,4]Triazolo[4,3-A]Pyridin-8-Yl)Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-12-19 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, HJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: NAP, HJG
 |
Crystal Structure Of Murine 11B- Hydroxysteroiddehydrogenase Complexed With 2-(3-(1-(4- Chlorophenyl)Cyclopropyl)-[1,2,4]Triazolo[4,3-A]Pyridin-8- Yl)Propan-2-Ol
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2018-12-19 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, HJG, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-12-19
Ligands: NAP, HJG, SO4
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[2-(4-Fluorophenyl)-2-Adamantyl]-1-(3-Methoxyazetidin-1-Yl)Ethanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8K4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8K4
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 1-(3-Hydroxyazetidin-1-Yl)-2-[(2S,5R)-2-(4-Fluorophenyl)-5-Methoxyadamantan-2-Yl]Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8K7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8K7
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[(1R,3S,5R,7S)-2-[4-(4-Fluorophenyl)Phenyl]-6-Hydroxyadamantan-2-Yl]-1-(3- Hydroxyazetidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KA
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-(2-Benzyl-6-Hydroxyadamantan-2-Yl)-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KD
 |
Crystal Structure Of 11Beta-Hsd1 Double Mutant (L262R, F278E) Complexed With 2-[(5R,7S)-6-Hydroxy-2-Phenyladamantan-2-Yl]-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One (Bms-816336)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KG
 |
Crystal Structure Of Murine 11Beta- Hydroxysteroiddehydrogenase Complexed With 2-[(5R,7S)-6-Hydroxy-2-Phenyladamantan-2-Yl]-1-(3-Hydroxyazetidin-1-Yl)Ethan-1-One (Bms-816336)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2017-11-01 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 8KG, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: NAP, 8KG, SO4
 |
Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With (1S,4S)-4-[8-(2-Fluorophenoxy)[1,2,4]Triazolo[4,3-A]Pyridin-3-Yl]Bicyclo[2.2.1]Heptan-1-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EO, CL
 |
Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With 3-[1-(4-Chlorophenyl)Cyclopropyl]-8-(2-Fluorophenoxy)[1,2,4]Triazolo[4,3-A]Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EN
 |
Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) In Complex With 3-[1-(4-Chlorophenyl)Cyclopropyl]-8-Cyclopropyl[1,2,4]Triazolo[4,3-A]Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-06-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, 1EQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: NAP, 1EQ
 |
Crystal Structure Of Dipeptidyl-Peptidase 4 (Cd26, Adenosine Deaminase Complexing Protein 2) (Dpp-Iv-Wt) Complex With Bms-767778 Aka 2-(3-(Aminomethyl)-4-(2,4- Dichlorophenyl)-2-Methyl-5-Oxo-5,7-Dihydro-6H-Pyrrolo[3,4- B]Pyridin-6-Yl)-N,N-Dimethylacetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-09-04 Classification: HYDROLASE Ligands: 1MD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: 1MD
 |
Crystal Structure Of Human Dpp-Iv In Complex With Bms-744891
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2013-09-04 Classification: HYDROLASE Ligands: 1WH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: 1WH
 |
Crystal Structure Of Human Dpp-Iv In Complex Withsa-(+)- Methyl2-(3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-2-Methyl- 7-Oxo-5H-Pyrrolo[3,4-B]Pyridin-6(7H)-Yl)Acetate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-02-29 Classification: hydrolase/hydrolase inhibitor Ligands: NAG, LGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-29
Ligands: NAG, LGE
 |
Crystal Structure Of 11B-Hsd1 Double Mutant (L262R, F278E) Complexed With 8-{[(2-Cyanopyridin-3-Yl)Methyl]Sulfanyl}-6-Hydroxy-3,4-Dihydro-1H-Pyrano[3,4-C]Pyridine-5-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-11-02 Classification: Oxidoreductase/Oxidoreductase Inhibitor Ligands: NAP, 07M, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: NAP, 07M, GOL
 |
Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, KXB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: NAG, KXB
 |
Crystal Structure Of Human Dpp-Iv In Complex With Sa-(+)-3-(Aminomethyl)-4-(2,4-Dichlorophenyl)-6-(2-Methoxyphenyl)- 2-Methyl-5H-Pyrrolo[3,4-B]Pyridin-7(6H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, KXA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: NAG, KXA
 |
X-Ray Crystal Structure Of Human Ppar Gamma With 2-(5-(3-(2-(5-Methyl-2-Phenyloxazol-4-Yl)Ethoxy)Benzyl)-2-Phenyl-2H-1,2,3-Triazol-4-Yl)Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2008-11-18 Classification: TRANSCRIPTION Ligands: ZAA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: ZAA