Search Count: 18
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Crystal Structure Of Btk Kinase Domain In Complex With Pirtobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: Y7W, SO4, GOL, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: Y7W, SO4, GOL, BTB
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Crystal Structure Of Btk C481S Kinase Domain In Complex With Pirtobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2023-03-01 Classification: TRANSFERASE/INHIBITOR Ligands: Y7W, SO4, GOL, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: Y7W, SO4, GOL, BTB
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Crystal Structure Of The Braf:Mek1 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2014-06-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACP, MG, 573, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: ACP, MG, 573, CL
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Crystal Structure Of Braf-V600E Bound To Gdc0879
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 29L, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 29L, CL
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Akt1 With Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-05-23 Classification: TRANSFERASE Ligands: ANP, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: ANP, MN
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Akt1 With Gdc0068
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-23 Classification: TRANSFERASE Ligands: 0RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-23
Ligands: 0RF
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Non-Oxime Pyrazole Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2011-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: SM7
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Spirocyclic Sulfonamides As Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: SM9
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMH
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMR
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Human B-Raf Kinase In Complex With A Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FOI
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Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FNI
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Crystal Structure Of Human B-Raf Kinase Domain In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP3
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Crystal Structure Of Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP4
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Furo[2,3-C]Pyridine-Based Indanone Oximes As Potent And Selective B-Raf Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-01-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: SM6
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Akt1 Kinase Domain With Pyrrolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: XM1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: XM1
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Crystal Structure Of C-Raf (Raf-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.00 Å Release Date: 2010-09-15 Classification: TRANSFERASE Ligands: SM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-15
Ligands: SM5
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Pyrazole-Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-08-19 Classification: TRANSFERASE Ligands: SM5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-08-19
Ligands: SM5