Search Count: 14
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Crystal Structure Of Orphan G Protein-Coupled Receptor 6 With Bound Inverse Agonist 3H
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2024-12-04 Classification: MEMBRANE PROTEIN Ligands: XY8, NA |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: XY8, NA
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Crystal Structure Of Orphan G Protein-Coupled Receptor 6 With Bound Cvn424
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:3.49 Å Release Date: 2024-12-04 Classification: MEMBRANE PROTEIN Ligands: X7T |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: X7T
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Crystal Structure Of Orphan G Protein-Coupled Receptor 6, Pseudoapo Form
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-12-04 Classification: MEMBRANE PROTEIN Ligands: OLC, P15, OLA, CLR |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: OLC, P15, OLA, CLR
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Cryo-Em Structure Of Gpr6-Gs-Nb35 Complex
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY Release Date: 2024-12-04 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Lama glama
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-04
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Crystal Structure Of 2-(3-Alkoxy-1-Azetidinyl) Quinolines As Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, GOL, 35E, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, GOL, 35E, ZN
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2-(3-Alkoxy-1-Azetidinyl) Quinolines As Novel Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, GOL, 35D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: ZN, SO4, GOL, 35D
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Hydroxyethylamine-Based Inhibitors Of Bace1: P1-P3 Macrocyclization Can Improve Potency, Selectivity, And Cell Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2013-07-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1QT
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Bace-1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2013-07-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1QU
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine-Macrocyclic Inhibitor 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-07-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1R8, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-03
Ligands: 1R8, GOL, SO4
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine-Macrocyclic Inhibitor 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-07-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, 1R6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-03
Ligands: IOD, 1R6, GOL
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine Inhibitor 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0K9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0K9, GOL
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Structure Of Bace-1 (Beta-Secretase) In Complex With N-((2S,3R)-1-(4-Fluorophenyl)-3-Hydroxy-4-((6'-Neopentyl-3',4'-Dihydrospiro[Cyclobutane-1,2'-Pyrano[2,3-B]Pyridin]-4'-Yl)Amino)Butan-2-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-10 Classification: HYDROLASE/Hydrolase Inhibitor Ligands: IOD, GOL, 0MP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: IOD, GOL, 0MP
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Structure Of Bace Bound To (S)-4-(3'-Methoxy-[1,1'-Biphenyl]-3-Yl)-1,4-Dimethyl-6-Oxotetrahydropyrimidin-2(1H)-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2012-10-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: H24, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: H24, TLA
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Structure Of Bace-1 (Beta-Secretase) In Complex With (2R)-N-((2S,3R)-1-(Benzo[D][1,3]Dioxol-5-Yl)-3-Hydroxy-4-((S)-6'-Neopentyl-3',4'-Dihydrospiro[Cyclobutane-1,2'-Pyrano[2,3-B]Pyridine]-4'-Ylamino)Butan-2-Yl)-2-Methoxypropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, GOL, 0KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-18
Ligands: IOD, GOL, 0KN