Search Count: 15
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Kras G13D Mutant In Complex With Gdp And Compound 6.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-06-03 Classification: ONCOPROTEIN Ligands: A1C3J, GDP, MG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: A1C3J, GDP, MG, PO4
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Kras G12V Mutant In Complex With Gdp And Compound 12.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2026-06-03 Classification: ONCOPROTEIN Ligands: MG, A1C3N, GDP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: MG, A1C3N, GDP, SO4
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Kras G12V Mutant In Complex With Gdp And Compound 8.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2026-06-03 Classification: ONCOPROTEIN Ligands: MG, A1C3O, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: MG, A1C3O, GDP
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Crystal Structure Of Phosphorylated Ret Tyrosine Kinase Domain Complexed With A Pyrrolo[2,3-D]Pyrimidine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.51 Å Release Date: 2022-01-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, 7QU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: CL, 7QU
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Leishmania Tarentolae Proteasome 20S Subunit Complexed With Lxe408
Organism: Leishmania donovani
Method: ELECTRON MICROSCOPY Release Date: 2020-08-26 Classification: HYDROLASE Ligands: N2E |
Organism: Leishmania donovani
Method: ELECTRON MICROSCOPY
Release Date: 2020-08-26
Ligands: N2E
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Leishmania Tarentolae Proteasome 20S Subunit Complexed With Lxe408 And Bortezomib
Organism: Leishmania donovani
Method: ELECTRON MICROSCOPY Release Date: 2020-08-26 Classification: HYDROLASE Ligands: BO2, N2E |
Organism: Leishmania donovani
Method: ELECTRON MICROSCOPY
Release Date: 2020-08-26
Ligands: BO2, N2E
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Dyrk1A Kinase Domain In Complex With A 6-Azaindole Derivative, Gnf2133.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2020-03-04 Classification: TRANSFERASE Ligands: Q8J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: Q8J
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Crystal Structure Of Phosphorylated Ret Tyrosine Kinase Domain Complexed With A Pyrazolo[1,5-A]Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-02-26 Classification: Transferase/Transferase Inhibitor Ligands: QX1, SO4, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-26
Ligands: QX1, SO4, CL, ACT
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-06-03 Classification: Transferase/Transferase inhibitor Ligands: 4EJ, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4EJ, GOL, CL
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2015-06-03 Classification: Transferase/Transferase inhibitor Ligands: 4EK, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4EK, SO4, GOL
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-06-03 Classification: Transfease/Transferase Inhibitor Ligands: 4F6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4F6, SO4
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Discovery Of A Selective Trk Inhibitor With Efficacy In Rodent Cancer Tumor Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, 0F4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: CL, 0F4
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Identification Of Novel Potent Bicyclic Peptide Deformylase Inhibitors
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2004-03-30 Classification: HYDROLASE Ligands: NI, GNR, GOL |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2004-03-30
Ligands: NI, GNR, GOL
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Hiv Integrase Core Domain Complexed With Tetraphenyl Arsonium
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2001-04-04 Classification: TRANSFERASE Ligands: SO4, CL, TTA |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2001-04-04
Ligands: SO4, CL, TTA
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Hiv Integrase Core Domain Complexed With A Derivative Of Tetraphenyl Arsonium.
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2001-04-04 Classification: TRANSFERASE Ligands: SO4, CL, TTO |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2001-04-04
Ligands: SO4, CL, TTO
