Search Count: 73
![]() |
Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-07-08 Classification: SIGNALING PROTEIN Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-08
Ligands: A1DEQ, A1DJL, GOL, SO4, DMS, EPE
![]() |
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: A1APL, DMS, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1APL, DMS, NA
![]() |
Crystal Structure Of Inhibitor 1 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: EDO, A1APO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: EDO, A1APO
![]() |
Crystal Structure Of Inhibitor Gne-6893 Bound To Hpk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2024-10-02 Classification: SIGNALING PROTEIN Ligands: MES, EDO, DMS, A1APR, NA, PEG, A1APQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: MES, EDO, DMS, A1APR, NA, PEG, A1APQ
![]() |
Crystal Structure Of A. Baumannii Guab Dcbs With Inhibitor G6 (3826)
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2024-09-18 Classification: OXIDOREDUCTASE Ligands: IMP, A1AUF |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2024-09-18
Ligands: IMP, A1AUF
![]() |
Co-Crystal Structure Of Phosphorylated Erk2 In Complex With Erk1/2 Inhibitor #16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-03-27 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: WAL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-27
Ligands: WAL
![]() |
Co-Crystal Structure Of Phosphorylated Erk2 In Complex With Erk1/2 Inhibitor #8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-03-27 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: W8U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-03-27
Ligands: W8U
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2YE
![]() |
Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F97, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: F97, EDO, MES
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2WI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2WI, SO4
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2TR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2TR
![]() |
Structure Of The Vps34 Kinase Domain With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
![]() |
Structure Of The Vps34 Kinase Domain With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: GOL, 7IK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: GOL, 7IK
![]() |
Structure Of The Vps34 Kinase Domain With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-11-24 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7IQ, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: 7IQ, GOL, NA
![]() |
Crystal Structure Of Braf In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: V5J, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: V5J, IOD
![]() |
Crystal Structure Of Braf In Complex With Inhibitor Gne-0749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VQP, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: VQP, CL
![]() |
Cdk2 In Complex With Cpd14 (5-Fluoro-4-(4-Methyl-5,6,7,8-Tetrahydro-4H-Pyrazolo[1,5-A]Azepin-3-Yl)-N-(5-(4-Methylpiperazin-1-Yl)Pyridin-2-Yl)Pyrimidin-2-Amine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-07-29 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: N14 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: N14
![]() |
Cdk6 In Complex With Cpd13 (R)-5-Fluoro-4-(4-Methyl-5,6,7,8-Tetrahydro-4H-Pyrazolo[1,5-A]Azepin-3-Yl)-N-(5-(4-Methylpiperazin-1-Yl)Pyridin-2-Yl)Pyrimidin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2020-07-29 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: N1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: N1A
![]() |
Cdk6 In Complex With Cpd24 N-(5-(6-Ethyl-2,6-Diazaspiro[3.3]Heptan-2-Yl)Pyridin-2-Yl)-5-Fluoro-4-(4-Methyl-5,6,7,8-Tetrahydro-4H-Pyrazolo[1,5-A]Azepin-3-Yl)Pyrimidin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-07-29 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: N1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: N1J
![]() |
Phosphorylated Erk2 With Amp-Pnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-07-31 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: ANP, MG
