Search Count: 13
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Crystal Structure Of Human Alk2 Kinase Domain With R206H Mutation In Complex With Rk783
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-06-25 Classification: SIGNALING PROTEIN Ligands: A1L4C, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: A1L4C, SO4
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2789
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: GOL, A1A29, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: GOL, A1A29, PO4
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2281
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: PO4, GOL, A1A3C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: PO4, GOL, A1A3C
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Crystal Structure Of The Acvr1 (Alk2) Kinase Domain In Complex With Inhibitor Cdd-2282
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-11-27 Classification: TRANSFERASE Ligands: A1A3D, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: A1A3D, PO4
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Braf In Complex With N-(4-Methyl-3-(1-Methyl-2-Oxo-2,3-Dihydro-1H-Benzo[D]Imidazol-5-Yl)Phenyl)-3-(Trifluoromethyl)Benzamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2019-10-23 Classification: transferase/transferase inhibitor Ligands: K7S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: K7S
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Braf In Complex With N-(3-(2-(2-Hydroxyethoxy)-6-Morpholinopyridin-4-Yl)-4-Methylphenyl)-2-(Trifluoromethyl)Isonicotinamide (Lxh254)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2019-09-04 Classification: transferase/transferase inhibitor Ligands: K81 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-04
Ligands: K81
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With Lsz102
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2018-04-04 Classification: HORMONE RECEPTOR Ligands: C6V, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: C6V, GOL
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-{4-[(1R)-2-(4-Fluorophenyl)-6-Hydroxy-1-Methy L-1,2,3,4- Tetrahydroisoquinolin-1-Yl]Phenyl}Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2017-03-29 Classification: HORMONE RECEPTOR Ligands: 77W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-29
Ligands: 77W
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Estrogen Receptor Alpha Ligand Binding Domain In Complex With (2E)-3-(4-{(1R)-6-Hydroxy-1-Methyl-2-[4-(Propan-2 -Yl)Phenyl]-1,2,3,4- Tetrahydroisoquinolin-1-Yl}Phenyl)Prop-2-Enoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-03-29 Classification: HORMONE RECEPTOR Ligands: 782 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-29
Ligands: 782
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Melk In Complex With Nvs-Melk1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-06-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-01
Ligands: 6BJ
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Melk In Complex With Nvs-Melk8A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2016-06-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-01
Ligands: 6BF
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Melk In Complex With Nvs-Melk8F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-06-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-01
Ligands: 6BE
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Melk In Complex With Nvs-Melk12B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2016-06-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6BB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-01
Ligands: 6BB
