Search Count: 35
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Protac-Mediated Complex Of Kras With Vhl/Elongin-B/Elongin-C/Cullin-2/Rbx1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.50 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: ZN, GDP, WYL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-12-06
Ligands: ZN, GDP, WYL
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Kras-G12C In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: GDP, MG, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, MG, WYU
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Crystal Structure Of Ligand Acbi3 In Complex With Kras G12D C118S Gdp And Pvhl:Elonginc:Elonginb Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2023-12-06 Classification: GENE REGULATION Ligands: PO4, WYL, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: PO4, WYL, GDP, MG
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Crystal Structure Of Compound 3 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: GDP, X4R, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, X4R, MG
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Crystal Structure Of Compound 4 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: X53, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: X53, GDP, MG
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Crystal Structure Of The Brd9 Bromodomain With Bi-7189
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-06-21 Classification: GENE REGULATION Ligands: M2O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: M2O
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Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
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Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
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Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
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Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
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Crystal Structure Of Compound 10 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IOD, IFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IOD, IFJ
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Crystal Structure Of Compound 6 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IFF
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Crystal Structure Of Compound 4 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IF8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IF8, ZN
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Crystal Structure Of Protac 5 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2022-09-07 Classification: LIGASE Ligands: IEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: IEI
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Crystal Structure Of The Bptf Bromodomain In Complex With Bi-7190
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.03 Å Release Date: 2022-08-31 Classification: PROTEIN BINDING Ligands: M1I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: M1I
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Crystal Structure Phgdh In Complex With Nadh And 3-Phosphoglycerate At 1.77 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: 3PG, NAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: 3PG, NAI
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Crystal Structure Of Phgdh In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: K4T, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: K4T, SO4
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Crystal Structure Of Phgdh In Complex With Compound 40
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K52
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Crystal Structure Of Phgdh In Complex With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K58
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Crystal Structure Of Phgdh In Complex With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K5N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K5N