Search Count: 21
![]() |
Crystal Structure Of Ack1 Kinase K161Q Mutant In Complex With The Selective Inhibitor (R)-9B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2023-03-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WTP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: WTP
![]() |
Structure Of Ack1 Kinase In Complex With A Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2022-02-09 Classification: TRANSFERASE/INHIBITOR Ligands: WTP, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-09
Ligands: WTP, CL
![]() |
Ddr1 Bound To Vx-680
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2018-12-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-05
Ligands: VX6
![]() |
Ddr1 Bound To Dasatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2018-12-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1N1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-05
Ligands: 1N1
![]() |
Src In Complex With Dna-Templated Macrocyclic Inhibitor Mc25B
Organism: Gallus gallus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-09-21 Classification: Transferase/transferase Inhibitor |
Organism: Gallus gallus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
![]() |
Crystal Structure Of The Activated Insulin Receptor Tyrosine Kinase Dimer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-03-25 Classification: TRANSFERASE Ligands: ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: ACP, MG
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domains Trapped In Trans-Phosphorylation Reaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-02-03 Classification: TRANSFERASE Ligands: MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-03
Ligands: MG, ACP
![]() |
Crystal Structure Of The Insulin-Like Growth Factor-1 Receptor Kinase In Complex With Pqip
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-07-29 Classification: TRANSFERASE Ligands: CA, D94 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-29
Ligands: CA, D94
![]() |
Crystal Structure Of Unphosphorylated Unactivated Wild Type Fgf Receptor 2 (Fgfr2) Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4
![]() |
Crystal Structure Of Tyrosine Phosphorylated Activated Fgf Receptor 2 (Fgfr2) Kinase Domain In Complex With Atp Analog And Substrate Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: MG, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic K659N Mutation Responsible For An Unclassified Craniosynostosis Syndrome.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic N549H Mutation Responsible For Crouzon Syndrome.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic E565G Mutation Responsible For Pfeiffer Syndrome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, MG, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic N549T Mutation Responsible For Pfeiffer Syndrome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, MG, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic K526E Mutation Responsible For Crouzon Syndrome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, MG, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, MG, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic K641R Mutation Responsible For Pfeiffer Syndrome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, ACP
![]() |
Crystal Structure Of Fgf Receptor 2 (Fgfr2) Kinase Domain Harboring The Pathogenic E565A Mutation Responsible For Pfeiffer Syndrome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, ACP
![]() |
Crystal Structure Of The C-Abl Kinase Domain In Complex With Pd173955
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2002-09-18 Classification: TRANSFERASE Ligands: P17, MES |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2002-09-18
Ligands: P17, MES
![]() |
Structure Of The Insulin-Like Growth Factor 1 Receptor Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2001-11-28 Classification: TRANSFERASE Ligands: ACP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2001-11-28
Ligands: ACP
![]() |
Crystal Structure Of The C-Abl Kinase Domain In Complex With Sti-571.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2001-04-18 Classification: TRANSFERASE Ligands: CL, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2001-04-18
Ligands: CL, STI
