Structural Entry Filters:

Search Count: 42

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9QXN image
Crystal Structure Of Wild-Type Egfr In Complex With The Reversible Inhibitor Sevabertinib (Bay 2927088)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.14 Å Release Date: 2025-10-15
Classification: TRANSFERASE
Ligands: SIN, CL, DMS, EDO, A1JBI

8ZU6 image
Solution Nmr Structure Of Pact D3 Homodimer

9FKR image
Kat6A In Complex With Small Molecule Inhibitor Bay-184
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.69 Å Release Date: 2024-11-06
Classification: TRANSFERASE
Ligands: ZN, A1IDR, EPE

8B8W image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.86 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q2X, GOL

8B8X image
Crystal Structure Of Pparg And Ncor2 With Sr10221, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.78 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: A8R

8B8Y image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q33

8B8Z image
Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.22 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q33

8B90 image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7D)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q1R

8B91 image
Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound Si-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.23 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q4O

8B92 image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound Si-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.66 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q5X, SO4

8B93 image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 15B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.21 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q8F

8B94 image
Crystal Structure Of Pparg And Ncor2 With Bay-5516, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q5O

8B95 image
Crystal Structure Of Pparg And Ncor2 With Bay-9683, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2022-12-28
Classification: TRANSCRIPTION
Ligands: Q4C

8AQM image
Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 6A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2022-11-09
Classification: TRANSCRIPTION
Ligands: O2O

8AQN image
Crystal Structure Of Pparg And Ncor2 With Bay-4931, An Inverse Agonist (Compound 6C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2022-11-09
Classification: TRANSCRIPTION
Ligands: O0U, GOL, CA

7KWE image
Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Dnmdp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2021-06-16
Classification: HYDROLASE
Ligands: X5M, MN, MG, ACT

7L27 image
Crystal Structure Of The Catalytic Domain Of Human Pde3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2021-06-16
Classification: HYDROLASE
Ligands: MN, MG, ACT, CA

7L28 image
Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Trequinsin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2021-06-16
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: XKG, MN, MG, ACT

7L29 image
Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Amp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.08 Å Release Date: 2021-06-16
Classification: HYDROLASE
Ligands: AMP, MN, MG, CA, ACT

7LRC image
Cryo-Em Of The Slfn12-Pde3A Complex: Pde3A Body Refinement
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