Search Count: 42
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Crystal Structure Of Wild-Type Egfr In Complex With The Reversible Inhibitor Sevabertinib (Bay 2927088)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-10-15 Classification: TRANSFERASE Ligands: SIN, CL, DMS, EDO, A1JBI |
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Solution Nmr Structure Of Pact D3 Homodimer
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2025-04-16 Classification: PROTEIN BINDING |
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Kat6A In Complex With Small Molecule Inhibitor Bay-184
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2024-11-06 Classification: TRANSFERASE Ligands: ZN, A1IDR, EPE |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q2X, GOL |
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Crystal Structure Of Pparg And Ncor2 With Sr10221, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: A8R |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound 7E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q33 |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 7D)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q1R |
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Crystal Structure Of Mutant Pparg (C313A) And Ncor2 With An Inverse Agonist (Compound Si-1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4O |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound Si-2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5X, SO4 |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 15B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q8F |
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Crystal Structure Of Pparg And Ncor2 With Bay-5516, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q5O |
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Crystal Structure Of Pparg And Ncor2 With Bay-9683, An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2022-12-28 Classification: TRANSCRIPTION Ligands: Q4C |
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Crystal Structure Of Pparg And Ncor2 With An Inverse Agonist (Compound 6A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-11-09 Classification: TRANSCRIPTION Ligands: O2O |
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Crystal Structure Of Pparg And Ncor2 With Bay-4931, An Inverse Agonist (Compound 6C)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-11-09 Classification: TRANSCRIPTION Ligands: O0U, GOL, CA |
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Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Dnmdp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-06-16 Classification: HYDROLASE Ligands: X5M, MN, MG, ACT |
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Crystal Structure Of The Catalytic Domain Of Human Pde3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-06-16 Classification: HYDROLASE Ligands: MN, MG, ACT, CA |
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Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Trequinsin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-06-16 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: XKG, MN, MG, ACT |
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Crystal Structure Of The Catalytic Domain Of Human Pde3A Bound To Amp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2021-06-16 Classification: HYDROLASE Ligands: AMP, MN, MG, CA, ACT |
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Cryo-Em Of The Slfn12-Pde3A Complex: Pde3A Body Refinement
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2021-06-09 Classification: HYDROLASE Ligands: MN, MG, X5M |




















