Search Count: 23
![]() |
The Discovery Of Novel, Potent And Highly Selective Inhibitors Of Inducible Nitric Oxide Synthase (Inos)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2014-10-08 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, YWO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: HEM, H4B, YWO
![]() |
Human Dpp1 In Complex With (2S)-2-Amino-N-((1S)-1-Cyano-2-(4- Phenylphenyl)Ethyl)Butanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-03-19 Classification: HYDROLASE Ligands: NAG, 6AO, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: NAG, 6AO, CL, GOL
![]() |
Human Dpp1 In Complex With (2S)-N-((1S)-1-Cyano-2-(4-(4-Cyanophenyl) Phenyl)Ethyl)Piperidine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-03-19 Classification: HYDROLASE Ligands: NAG, GDI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: NAG, GDI, CL
![]() |
Human Dpp1 In Complex With 4-Amino-N-((1S)-1-Cyano-2-(4-(4- Cyanophenyl)Phenyl)Ethyl)Tetrahydropyran-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-03-19 Classification: HYDROLASE Ligands: NAG, U6B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: NAG, U6B, CL
![]() |
Human Dpp1 In Complex With (2S,4S)-N-((1S)-1-Cyano-2-(4-(4- Cyanophenyl)Phenyl)Ethyl)-4-Hydroxy-Piperidine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-03-19 Classification: HYDROLASE Ligands: NAG, W2C, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: NAG, W2C, CL
![]() |
The Discovery Of Novel, Potent And Highly Selective Inhibitors Of Inducible Nitric Oxide Synthase (Inos)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-04-13 Classification: OXIDOREDUCTASE Ligands: SO4, GOL, A54, HEM, H4B |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-04-13
Ligands: SO4, GOL, A54, HEM, H4B
![]() |
Murine Inos Dimer With Heme, Pterin And Inhibitor Ar-C120011
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, XXZ |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, XXZ
![]() |
Murine Inos Dimer With Inhibitor 4-Map Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, BVF |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, BVF
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C130232
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: BOG, SO4, AT6, HEM, H4B, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: BOG, SO4, AT6, HEM, H4B, EDO
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C132283
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: BOG, SO4, HEM, H4B, A11 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: BOG, SO4, HEM, H4B, A11
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C125813
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, AS3 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, AS3
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C124355
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, A55 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, A55
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C118901
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, 1A2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, 1A2
![]() |
Structure Of Human Inosox With Inhibitor Ar-C95791
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: ZN, HEM, H4B, AT2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: ZN, HEM, H4B, AT2
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C94864
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: SO4, ZN, HEM, H4B, B2 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: SO4, ZN, HEM, H4B, B2
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C95791
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: ZN, HEM, H4B, AT2, EDO |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: ZN, HEM, H4B, AT2, EDO
![]() |
Structure Of Bovine Enos Oxygenase Domain With Inhibitor Ar-C95791
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: ZN, HEC, AT2 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: ZN, HEC, AT2
![]() |
Structure Of Murine Inos Oxygenase Domain With Inhibitor Ar-C102222
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: SO4, HEM, HBI, B14 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: SO4, HEM, HBI, B14
![]() |
Structure Of Inhibited Human Enos Oxygenase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEC, ZN, 327, MPD, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEC, ZN, 327, MPD, CL
![]() |
Structure Of Inhibited Murine Inos Oxygenase Domain
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-10-07 Classification: OXIDOREDUCTASE Ligands: HEM, H4B, 328, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2008-10-07
Ligands: HEM, H4B, 328, SO4
