Search Count: 15
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Human P300 Complexed With A Proline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C0C
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Human P300 Complexed With A Glycine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C3I, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C3I, ACT
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Human P300 Complexed With An Azaindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ETL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ETL
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Alpha-1 Antitrypsin C232S Complexed With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-04-07 Classification: UNKNOWN FUNCTION Ligands: GOL, UL2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: GOL, UL2
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Alpha-1 Antitrypsin (C232S) Complexed With Cmpd 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2021-04-07 Classification: UNKNOWN FUNCTION Ligands: UKZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: UKZ, GOL
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Alpha 1-Antitrypsin (C232S) Complexed With Gsk716
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-03-10 Classification: PROTEIN BINDING Ligands: R7Z, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: R7Z, SO4
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Crystal Structure Of Steptococcus Pneumoniae Undecaprenyl Pyrophosphate Synthase (Upps)
Organism: Streptococcus pneumoniae serotype 4 (strain atcc baa-334 / tigr4)
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-07-20 Classification: TRANSFERASE |
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Crystal Structure Of Steptococcus Pneumoniae Undecaprenyl Pyrophosphate Synthase (Upps) With Farnesyl Diphosphate
Organism: Streptococcus pneumoniae serotype 4 (strain atcc baa-334 / tigr4)
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2016-07-20 Classification: TRANSFERASE Ligands: FPP |
Organism: Streptococcus pneumoniae serotype 4 (strain atcc baa-334 / tigr4)
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: FPP
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Crystal Structure Of Steptococcus Pneumoniae Undecaprenyl Pyrophosphate Synthase (Upps) In Complex With ~{N}-(3-Azanyl-3-Oxidanylidene-Propyl)-5-(1-Benzothiophen-5-Yl)-1-(Phenylmethyl)-~{N}-[(4-Propan-2-Yloxyphenyl)Methyl]Pyrazole-4-Carboxamide
Organism: Streptococcus pneumoniae serotype 4 (strain atcc baa-334 / tigr4)
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2016-07-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6TC |
Organism: Streptococcus pneumoniae serotype 4 (strain atcc baa-334 / tigr4)
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: 6TC
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X-Ray Crystal Structure Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A 2-Aryl Benzimidazole Compound And An Internal Aldimine Linked Plp Cofactor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2016-05-04 Classification: TRANSFERASE Ligands: PLP, EL2, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: PLP, EL2, CL, EDO, GOL
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X-Ray Crystal Structure At 1.61A Resolution Of Human Mitochondrial Branched Chain Aminotransferase (Bcatm) Complexed With A Biphenyl Pyrrolidine Ether Compound And An Internal Aldimine Linked Plp Cofactor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: PLP, EL1, CL, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: PLP, EL1, CL, EDO, DMS
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Crystal Structure Of Gantenerumab Fab Fragment In Complex With Abeta 1-11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-12 Classification: IMMUNE SYSTEM Ligands: NAG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: NAG, SO4
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Encoded Library Technology As A Source Of Hits For The Discovery And Lead Optimization Of A Potent And Selective Class Of Bactericidal Direct Inhibitors Of Mycobacterium Tuberculosis Inha
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-02-12 Classification: TRANSFERASE Ligands: KV1, NAD |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: KV1, NAD
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Crystal Structure Of Aurora A In Complex With Tpx2 And Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2009-08-04 Classification: TRANSFERASE Ligands: 2JZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-08-04
Ligands: 2JZ
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The Complex Structure Of The Map Kinase P38/Compound 14B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2009-08-04 Classification: TRANSFERASE Ligands: 5JZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-08-04
Ligands: 5JZ
