Search Count: 18
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Bace1 In Complex With (S)-5-(3-Chloro-5-(5-(Prop-1-Yn-1-Yl)Pyridin-3-Yl)Thiophen-2-Yl)-2,5-Dimethyl-1,2,4-Thiadiazinan-3-Iminium 1,1-Dioxide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66J
 |
Bace1 In Complex With 4-(3-(Furan-2-Carboxamido)Phenyl)-1-Methyl-5-Oxo-4-Phenylimidazolidin-2-Iminium
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: TLA, 66H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: TLA, 66H
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Bace1 In Complex With (R)-N-(3-(3-Amino-2,5-Dimethyl-1,1-Dioxido-5,6-Dihydro-2H-1,2,4-Thiadiazin-5-Yl)-4-Fluorophenyl)-5-Fluoropicolinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 66F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 66F
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With N-(N-(4-Amino-3,5- Dichlorobenzyl)Carbamimidoyl)-3-(4-Methoxyphenyl)-5- Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VA, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VA, IOD
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Db-Mut) Complex With N-(N-(4- Acetamido-3-Chloro-5-Methylbenzyl)Carbamimidoyl)-3-(4- Methoxyphenyl)-5-Methyl-4-Isothiazolecarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-10 Classification: HYDROLASE/INHIBITOR Ligands: 0VB, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0VB, IOD
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Eval Processed Hewl, Cisplatin Aqueous Glycerol
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: GOL
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Eval Processed Hewl, Cisplatin Aqueous Paratone
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: MEB |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: MEB
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Eval Processed Hewl, Carboplatin Aqueous Glycerol
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: GOL
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Eval Processed Hewl, Carboplatin Aqueous Paratone
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: CL, MEB |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: CL, MEB
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Eval Processed Hewl, Carboplatin Dmso Glycerol
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: QPT, DMS, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: QPT, DMS, GOL
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Eval Processed Hewl, Carboplatin Dmso Paratone
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: QPT, DMS |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: QPT, DMS
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Eval Processed Hewl, Cisplatin Dmso Paratone Ph 6.5
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: CPT, DMS |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: CPT, DMS
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Eval Processed Hewl, Cisplatin Dmso Nag Silicone Oil
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-04-25 Classification: HYDROLASE Ligands: CPT, DMS |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: CPT, DMS
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3R)-3-Acetamido-3-Isobutyl-2-Oxo-1-Pyrrolidinyl)-N-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-2-(1,2,3,4-Tetrahydro-3-Isoquinolinyl)Ethyl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2011-09-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-07
Ligands: PB8
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With Bms-693391 Aka (2S)-2-((3R)-3-Acetamido-3-Isobutyl-2-Oxo-1-Pyrrolidinyl)-N-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-2-((2R,4R)-4-Propoxy-2-Pyrrolidinyl)Ethyl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PB0
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With (2S)-2-((3S)-3-(Acetylamino)-3-(Butan-2-Yl)-2-Oxopyrrolidin-1-Yl)-N-((2S,3R)-3-Hydroxy-4-((3-Methoxybenzyl)Amino)-1-Phenylbutan-2-Yl)-4-Phenylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: PB7, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PB7, IOD
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With Bms-655295 Aka N~3~-((1S,2R)-1- Benzyl-2-Hydroxy-3-((3-Methoxybenzyl)Amino)Propyl)-N~1~, N~1~-Dibutyl-1H-Indole-1,3-Dicarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3HF, IOD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: 3HF, IOD, GOL
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Crystal Structure Of Beta-Site App-Cleaving Enzyme 1 (Bace-Wt) Complex With Bms-681889 Aka N~1~-Butyl-5-Cyano- N~3~-((1S,2R)-1-(3,5-Difluorobenzyl)-2-Hydroxy-3-((3- Methoxybenzyl)Amino)Propyl)-N~1~-Methyl-1H-Indole-1,3- Dicarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2011-04-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3HH, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: 3HH, SO4, GOL