Search Count: 23
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Crystal Structure Of Nedd4 Hect Domain In Complex With Norclomipramine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2025-06-04 Classification: LIGASE Ligands: EDO, A1ITH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-04
Ligands: EDO, A1ITH
 |
Crystal Structure Of Nedd4 Hect Domain In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2025-06-04 Classification: LIGASE Ligands: A1ITT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-04
Ligands: A1ITT
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 2-[3-{4-Chloro-3-[(4-Chlorophenyl)Ethynyl]Phenyl}-1-(3-Morpholin-4-Ylpropyl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl]-2-Oxoethanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2020-06-03 Classification: OXIDOREDUCTASE Ligands: N4K, FAD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: N4K, FAD, GOL
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W0
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W3
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Thieno[3,2-B]Pyrrole-5-Carboxamides As Novel Reversible Inhibitors Of Histone Lysine Demethylase Kdm1A/Lsd1: Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6W1
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Methyl-N-[4-[[4-(1-Methylpiperidin-4-Yl)Oxyphenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X3
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Structure Of The Kdm1A/Corest Complex With The Inhibitor 4-Ethyl-N-[3-(Methoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]Thieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, GOL, 6X0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, GOL, 6X0
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Structure Of The Kdm1A/Corest Complex With The Inhibitor N-[3-(Ethoxymethyl)-2-[[4-[[(3R)-Pyrrolidin-3-Yl]Methoxy]Phenoxy]Methyl]Phenyl]-4-Methylthieno[3,2-B]Pyrrole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2017-02-22 Classification: OXIDOREDUCTASE Ligands: FAD, 6X5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: FAD, 6X5, GOL
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Lsd1(Kdm1A)-Corest In Complex With Z-Pro Derivative Of Mc2580
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-02-25 Classification: OXIDOREDUCTASE Ligands: FAD, M8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-25
Ligands: FAD, M8A
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Lsd1(Kdm1A)-Corest In Complex With 1-Benzyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D69 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D69
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Lsd1(Kdm1A)-Corest In Complex With 1-Ethyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D70 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D70
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Lsd1(Kdm1A)-Corest In Complex With 1-Methyl-Tranylcypromine (1R,2S)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D73 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D73
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Lsd1(Kdm1A)-Corest In Complex With 1-Methyl-Tranylcypromine (1S,2R)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D51 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D51
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Lsd1(Kdm1A)-Corest In Complex With 1-Phenyl-Tranylcypromine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2014-09-10 Classification: TRANSCRIPTION Ligands: D52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-10
Ligands: D52
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Optimisation Of 6,6-Dimethyl Pyrrolo 3,4-C Pyrazoles: Identification Of Pha-793887, A Potent Cdk Inhibitor Suitable For Intravenous Dosing
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-02-23 Classification: CELL CYCLE Ligands: SO4, 889 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: SO4, 889
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Structure Of Cdk2-Cyclin A With A Pyrazolo(4,3-H) Quinazoline-3- Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-02-23 Classification: TRANSFERASE Ligands: WXV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-02-23
Ligands: WXV, SO4
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Structure Of Cdk2-Cyclin A With Pha-848125
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P48, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P48, SO4
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Structure Of Cdk2-Cyclin A Complexed With 8-Anilino-1-Methyl-4,5-Dihydro- 1H-Pyrazolo[4,3-H] Quinazoline-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-07-28 Classification: TRANSFERASE Ligands: P49, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-07-28
Ligands: P49, SO4
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Structure Of Hsp90 Bound With A Noval Fragment.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-06-30 Classification: CHAPERONE Ligands: MOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-06-30
Ligands: MOJ