Search Count: 14
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Discovery Of The First Orally Bioavailable Adamts7 Inhibitor Bay-9835
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2024-02-21 Classification: HYDROLASE Ligands: ZN, CA, A1H07, PEG, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: ZN, CA, A1H07, PEG, CL
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Coagulation Factor Xi Protease Domain In Complex With Active Site Inhibitor Asundexian
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2023-09-13 Classification: BLOOD CLOTTING Ligands: QV3, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-13
Ligands: QV3, CIT
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Coagulation Factor Xi Protease Domain In Complex With Active Site Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2023-09-13 Classification: BLOOD CLOTTING Ligands: GOL, QVI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-13
Ligands: GOL, QVI
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Coagulation Factor Xi Protease Domain In Complex With Active Site Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-09-13 Classification: BLOOD CLOTTING Ligands: QVO, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-13
Ligands: QVO, CIT, GOL
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Coagulation Factor Xi Protease Domain In Complex With Active Site Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2023-09-13 Classification: BLOOD CLOTTING Ligands: QW0, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-13
Ligands: QW0, CIT, GOL
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Coagulation Factor Xi Protease Domain In Complex With Active Site Inhibitor 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2023-09-13 Classification: BLOOD CLOTTING Ligands: QW6, CIT, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-13
Ligands: QW6, CIT, TRS
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X-Ray Structure Of Pde9A In Complex With Inhibitor 13A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2022-12-28 Classification: HYDROLASE Ligands: ZN, MG, NA, R4I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: ZN, MG, NA, R4I
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-08-03 Classification: HYDROLASE Ligands: NAG, IUY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: NAG, IUY
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-03 Classification: HYDROLASE Ligands: VBM, MES, MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: VBM, MES, MLI
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-08-03 Classification: HYDROLASE Ligands: NAG, IUL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: NAG, IUL
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: NAG, JJD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: NAG, JJD
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: JJS, NAG, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: JJS, NAG, EPE
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: NAG, JJX, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: NAG, JJX, DMS
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Crystal Structure Of Human Neutrophil Elastase In Complex With A Dihydropyrimidone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-08-19 Classification: HYDROLASE Ligands: JJV, MES, XPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-19
Ligands: JJV, MES, XPE
