Search Count: 36
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X-Ray Co-Crystal Structure Of Compound 7 With Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-12-11 Classification: APOPTOSIS/INHIBITOR Ligands: Q57 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: Q57
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X-Ray Co-Crystal Structure Of Compound 5 With Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-12-11 Classification: APOPTOSIS/INHIBITOR Ligands: Q54 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-11
Ligands: Q54
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Co-Crystal Structure Of Compound 1 Bound To Human Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2019-12-04 Classification: APOPTOSIS/INHIBITOR Ligands: Q4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q4D
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X-Ray Co-Crystal Structure Of Compound 20 With Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2019-12-04 Classification: APOPTOSIS/INHIBITOR Ligands: Q4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q4S
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X-Ray Co-Crystal Structure Of Compound 10 Bound To Human Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-04 Classification: APOPTOSIS/INHIBITOR Ligands: Q4V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q4V
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X-Ray Co-Crystal Structure Of Compound 8 Bound To Human Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2019-12-04 Classification: APOPTOSIS/INHIBITOR Ligands: Q4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q4Y
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X-Ray Co-Crystal Structure Of Compound 3 Bound To Human Mcl-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2019-12-04 Classification: APOPTOSIS/INHIBITOR Ligands: Q51 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q51
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Glucocorticoid Receptor In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2018-10-03 Classification: TRANSCRIPTION Ligands: HJ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: HJ4
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Crystal Structure Of Human Pi3K-Gamma In Complex With Quinoline-Containing Inhibitor 5G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-06-21 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 6RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: SO4, 6RF
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Crystal Structure Of Human Pi3K-Gamma In Complex With Benzimidazole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 5MT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5MT
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Crystal Structure Of Compound 16 Bound To Mdm2(17-111), {(3R,5R,6S)-5-(3-Chlorophenyl)-6-(4-Chlorophenyl)-1-[(1S)-1-Cyclopropyl-2-(Pyrrolidin-1-Ylsulfonyl)Ethyl]-3-Methyl-2-Oxopiperidin-3-Yl}Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-05-06 Classification: Ligase/Ligase inhibitor Ligands: 35T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 35T
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Crystal Structure Of Human Pi3K-Gamma In Complex With (S)-N-(1-(7-Fluoro-2-(Pyridin-2-Yl)Quinolin-3-Yl)Ethyl)-9H-Purin-6-Amine Amg319 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VC
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Crystal Structure Of Human Pi3K-Gamma In Complex With Phenylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(3-Fluorophenyl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VD
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Crystal Structure Of Human Pi3K-Gamma In Complex With Pyridinylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(2-Methylpyridin-3-Yl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VE, GOL
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Co-Crystal Structure Of Mdm2 In Complex With Am-7209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2014-12-03 Classification: LIGASE/LIGASE INHIBITOR Ligands: 3UD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: 3UD, SO4
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Crystal Structure Of A Cdk6/Vcyclin Complex With Inhibitor Bound
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-08-06 Classification: TRANSFERASE/CELL CYCLE/INHIBITOR Ligands: 24V |
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: 24V
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Co-Crystal Structure Of Mdm2 (17-111) With Compound 16, {(3R,5R,6S)-5-(3-Chlorophenyl)-6-(4-Chlorophenyl)-1-[(1S)-1-(6-Cyclopropylpyridin-2-Yl)Propyl]-3-Methyl-2-Oxopiperidin-3-Yl}Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-07-16 Classification: Ligase/Ligase inhibitor Ligands: 35S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-16
Ligands: 35S
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Crystal Structure Of Retinol-Binding Protein 4 (Rbp4)In Complex With A Non-Retinoid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-07-02 Classification: PROTEIN BINDING Ligands: 2RY, EDO, CL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-02
Ligands: 2RY, EDO, CL, PEG
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Crystal Structure Of Retinol-Binding Protein 4 (Rbp4) In Complex With A Non-Retinoid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-02 Classification: TRANSPORT PROTEIN Ligands: 2WL, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-02
Ligands: 2WL, PO4, EDO
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Co-Crystal Structure Of Mdm2(17-111) In Complex With Compound 48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-04-02 Classification: ligase/ligase inhibitor Ligands: 2TZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2TZ
