Search Count: 22
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Glucocorticoid Receptor In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2018-10-03 Classification: TRANSCRIPTION Ligands: HJ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: HJ4
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Crystal Structure Of Human Pi3K-Gamma In Complex With Quinoline-Containing Inhibitor 5G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-06-21 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 6RF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-21
Ligands: SO4, 6RF
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Crystal Structure Of Human Pi3K-Gamma In Complex With Benzimidazole Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 5MT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5MT
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Crystal Structure Of Compound 16 Bound To Mdm2(17-111), {(3R,5R,6S)-5-(3-Chlorophenyl)-6-(4-Chlorophenyl)-1-[(1S)-1-Cyclopropyl-2-(Pyrrolidin-1-Ylsulfonyl)Ethyl]-3-Methyl-2-Oxopiperidin-3-Yl}Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2015-05-06 Classification: Ligase/Ligase inhibitor Ligands: 35T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 35T
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Crystal Structure Of Human Pi3K-Gamma In Complex With (S)-N-(1-(7-Fluoro-2-(Pyridin-2-Yl)Quinolin-3-Yl)Ethyl)-9H-Purin-6-Amine Amg319 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VC
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Crystal Structure Of Human Pi3K-Gamma In Complex With Phenylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(3-Fluorophenyl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VD
 |
Crystal Structure Of Human Pi3K-Gamma In Complex With Pyridinylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(2-Methylpyridin-3-Yl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VE, GOL
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Co-Crystal Structure Of Mdm2 In Complex With Am-7209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2014-12-03 Classification: LIGASE/LIGASE INHIBITOR Ligands: 3UD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: 3UD, SO4
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Crystal Structure Of A Cdk6/Vcyclin Complex With Inhibitor Bound
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-08-06 Classification: TRANSFERASE/CELL CYCLE/INHIBITOR Ligands: 24V |
Organism: Saimiriine herpesvirus 2, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: 24V
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Co-Crystal Structure Of Mdm2(17-111) In Complex With Compound 48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-04-02 Classification: ligase/ligase inhibitor Ligands: 2TZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2TZ
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U0, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 47
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U1
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Co-Crystal Structure Of Mdm2 With Inhbitor Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U5, SO4
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Co-Crystal Structure Of Mdm2 With Inhbitor Compound 46
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U6, SO4
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 49
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: LIGASE/LIGASE INHIBITOR Ligands: 2U7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 2U7
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Co-Crystal Structure Of Mdm2 With Inhibitor Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-03-19 Classification: ligase/ligase inhibitor Ligands: 2TW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: 2TW
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Co-Crystal Structure Of Mdm2 (17-111) In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-02-19 Classification: ligase/ligase inhibitor Ligands: 2SW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-19
Ligands: 2SW, SO4
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Crystal Structure Of Nik With 11-Bromo-5,6,7,8-Tetrahydropyrimido[4',5':3,4]Cyclohepta[1,2-B]Indol-2-Amine (T28)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-04-17 Classification: Transferase/Transferase Inhibitor Ligands: T28 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: T28
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Crystal Structure Of Nik With Compound 4-{3-[2-Amino-5-(2-Methoxyethoxy)Pyrimidin-4-Yl]-1H-Indol-5-Yl}-2-Methylbut-3-Yn-2-Ol (13V)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-04-17 Classification: Transferase/Transferase Inhibitor Ligands: 13V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: 13V
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Crystal Structure Of Pi3K-Gamma In Complex With Quinoline-Indoline Inhibitor 24F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2012-10-24 Classification: Transferase/Inhibitor Ligands: SO4, FJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: SO4, FJY