Search Count: 22
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Yeast Sdd1 Disome With Mbf1
Organism: Saccharomyces cerevisiae
Method: ELECTRON MICROSCOPY Release Date: 2024-12-04 Classification: RIBOSOME Ligands: MG, ZN, K, SPD |
Organism: Saccharomyces cerevisiae
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-04
Ligands: MG, ZN, K, SPD
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Structures Of Rev1 Ubm2 Domain Complex With Ubiquitin And With The First Small-Molecule That Inhibits The Rev1 Ubm2-Ubiquitin Interaction
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2018-06-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2018-06-27
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Rev1 Ubm2 Domain Complex With Ubiquitin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2018-06-20 Classification: PROTEIN BINDING Ligands: NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: NI
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Cct068127 In Complex With Cdk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2017-12-20 Classification: CELL CYCLE/INHIBITOR Ligands: 8QT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: 8QT
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Crystal Structure Of Prmt5:Mep50 In Complex With Mta And H4 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2016-02-24 Classification: TRANSFERASE/PROTEIN BINDING Ligands: MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: MTA
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Structure Of Aurora-A Bound To An Imidazopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-09-22 Classification: TRANSFERASE Ligands: ASH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: ASH
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Structure Of Aurora-A Bound To A Selective Imidazopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2010-09-22 Classification: TRANSFERASE Ligands: A0H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: A0H
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Aurora-A Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-07-07 Classification: TRANSFERASE Ligands: SO4, X6D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-07
Ligands: SO4, X6D
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Aurora-A Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2010-07-07 Classification: TRANSFERASE Ligands: YM4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-07
Ligands: YM4
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2GJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2GJ
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4,5 Diaryl Isoxazole Hsp90 Chaperone Inhibitors: Potential Therapeutic Agents For The Treatment Of Cancer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2007-12-11 Classification: CHAPERONE Ligands: 2EQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-12-11
Ligands: 2EQ
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Inhibition Of The Hsp90 Molecular Chaperone In Vitro And In Vivo By Novel, Synthetic, Potent Resorcinylic Pyrazole, Isoxazole Amide Analogs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2007-04-24 Classification: CHAPERONE Ligands: MG, SO4, 2GG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-24
Ligands: MG, SO4, 2GG
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Structure Of Camp-Dependent Protein Kinase Complexed With Isoquinoline-5-Sulfonic Acid (2-(2-(4-Chlorobenzyloxy)Ethylamino) Ethyl)Amide
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2005-11-02 Classification: TRANSFERASE/INHIBITOR Ligands: I5S |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-02
Ligands: I5S
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Structure Of Camp-Dependent Protein Kinase Complexed With (4R,2S)-5'-(4-(4-Chlorobenzyloxy)Pyrrolidin-2-Ylmethanesulfonyl)Isoquinoline
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-11-02 Classification: TRANSFERASE/INHIBITOR Ligands: CQP |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-02
Ligands: CQP
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Structure Of A Hsp90 Inhibitor Bound To The N-Terminus Of Yeast Hsp90.
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2005-09-29 Classification: CHAPERONE Ligands: CT5 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2005-09-29
Ligands: CT5
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Structure Of A Hsp90 Inhibitor Bound To The N-Terminus Of Yeast Hsp90.
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-09-29 Classification: CHAPERONE Ligands: KJ2 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2005-09-29
Ligands: KJ2
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Synthesis And Activity Of N-Axyl Azacyclic Urea Hiv-1 Protease Inhibitors With High Potency Against Multiple Drug Resistant Viral Strains.
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-09-20 Classification: HYDROLASE Ligands: AAU |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2005-09-20
Ligands: AAU
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Novel, Potent Small Molecule Inhibitors Of The Molecular Chaperone Hsp90 Discovered Through Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2005-06-02 Classification: CHAPERONE Ligands: BSM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-02
Ligands: BSM
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Novel, Potent Small Molecule Inhibitors Of The Molecular Chaperone Hsp90 Discovered Through Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-06-02 Classification: CHAPERONE Ligands: CT5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-02
Ligands: CT5
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Crystal Structure Of A Fyve-Type Domain From Caspase Regulator Carp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2004-12-28 Classification: METAL BINDING PROTEIN Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-12-28
Ligands: ZN
