Search Count: 15
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Cryoem Structure Of Nlrp3 Nacht Domain In Complex With G2394
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2022-11-02 Classification: HYDROLASE Ligands: MG, ADP, WTN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2022-11-02
Ligands: MG, ADP, WTN
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Structure-Guided Optimization Of A Novel Class Of Ask1 Inhibitors With Increased Sp3 Character And An Exquisite Selectivity Profile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2020-08-12 Classification: METAL BINDING PROTEIN Ligands: V3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: V3S
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: 79D, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: 79D, ZN
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Crystal Structure Of Plk1 In Complex With A Novel 5,6-Dihydroimidazolo[1,5-F]Pteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: ZN, 79C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: ZN, 79C
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Potent, Reversible Metap2 Inhibitors Via Fragment Based Drug Discovery
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-05-25 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MN, DMS, EDO, 6KP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, DMS, EDO, 6KP
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Potent, Reversible Metap2 Inhibitors Via Fbdd
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-05-25 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MN, GOL, DMS, 6KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, DMS, 6KO
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Potent, Reversible Metap2 Inhibitors Via Fbdd
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-05-25 Classification: Hydrolase4/Hydrolase Inhibitor Ligands: MN, SO4, 6KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, SO4, 6KN
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Braf In Complex With Raf265
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.17 Å Release Date: 2015-09-09 Classification: TRANSFERASE Ligands: 55J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: 55J
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Crystal Structure Of Hsp90-Alpha N-Domain Bound To The Inhibitor Nvp-Hsp990
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-11-26 Classification: CHAPERONE/INHIBITOR Ligands: 3JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: 3JC
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Crystal Structure Of Hsp90-Alpha N-Domain Bound To The Inhibitor Nvp-Hsp990
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-11-19 Classification: CHAPERONE Ligands: 990 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: 990
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Pim1 Complexed With A Phenylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HV
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HW, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HW, GOL
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Pim1 Complexed With A Pyridylcarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-06
Ligands: 2HX
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Crystal Structure Of Plk1 In Complex With A Pyrimidodiazepinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J3, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 1J3, ZN, ACT
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Crystal Structure Of Plk1 In Complex With Tak-960
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, ACT, 1J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: ZN, ACT, 1J4