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8FRL image
Acinetobacter Baylyi Lptb2Fg Bound To Lipopolysaccharide And A Macrocyclic Peptide
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: Y75, JSG, LMT

8FRM image
Acinetobacter Baylyi Lptb2Fg Bound To Lipopolysaccharide.
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: JSG

8FRN image
Acinetobacter Baylyi Lptb2Fg Bound To Lipopolysaccharide And Zosurabalpin
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: JSG, VB6, LMT

8FRO image
Acinetobacter Baylyi Lptb2Fg Bound To Lipopolysaccharide And A Macrocyclic Peptide
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: JSG, MG3

8FRP image
Acinetobacter Baylyi Lptb2Fgc
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT

8UFG image
Acinetobacter Baylyi Lptb2Fg Bound To Acinetobacter Baylyi Lipopolysaccharide
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: LMT, WJR

8UFH image
Acinetobacter Baylyi Lptb2Fg Bound To Acinetobacter Baylyi Lipopolysaccharide And A Macrocyclic Peptide
Organism: Acinetobacter baylyi adp1
Method: ELECTRON MICROSCOPY
Release Date: 2024-01-03
Classification: LIPID TRANSPORT
Ligands: WJW, Y75

5S9L image
Autotaxin, 4-[3-Oxo-3-(2-Oxo-2,3-Dihydro-Benzooxazol-6-Yl)-Propyl]-Piperazine-1-Carboxylic Acid 3,5-Dichloro-Benzyl Ester, 1.90A, P212121, Rfree=19.1%
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2022-04-13
Classification: HYDROLASE
Ligands: CA, K, ACT, 6ZO, ZN, NA

5S9M image
Autotaxin, (3,5-Dichlorophenyl)Methyl (3As,8Ar)-2-(1H-Benzotriazole-5-Carbonyl)-1,3,3A,4,5,7,8,8A-Octahydropyrrolo[3,4-D]Azepine-6-Carboxylate, 1.80A, P212121, Rfree=21.1%
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2022-04-13
Classification: HYDROLASE
Ligands: YV1, ACT, PG4, ZN, CA, CL, NA

5S9N image
Autotaxin, [4-(Trifluoromethoxy)Phenyl]Methyl (3As,6As)-2-(1H-Benzotriazole-5-Carbonyl)-1,3,3A,4,6,6A-Hexahydropyrrolo[3,4-C]Pyrrole-5-Carboxylate, 1.80A, P212121, Rfree=23.3%
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.80 Å Release Date: 2022-04-13
Classification: HYDROLASE
Ligands: YVS, ZN, CA, CL, NA

5LP4 image
Penicillin-Binding Protein (Pbp2) From Helicobacter Pylori
Organism: Helicobacter pylori (strain atcc 700392 / 26695)
Method: X-RAY DIFFRACTION
Resolution:3.03 Å Release Date: 2017-08-23
Classification: HYDROLASE/ANTIBIOTIC
Ligands: SO4

5LP5 image
Complex Between Penicillin-Binding Protein (Pbp2) And Mrec From Helicobacter Pylori
Organism: Helicobacter pylori (strain atcc 700392 / 26695)
Method: X-RAY DIFFRACTION
Resolution:2.74 Å Release Date: 2017-08-23
Classification: HYDROLASE/ANTIBIOTIC

5SVA image
Mediator-Rna Polymerase Ii Pre-Initiation Complex
Method: ELECTRON MICROSCOPY
Release Date: 2016-09-28
Classification: TRANSCRIPTION, TRANSFERASE/DNA
Ligands: ZN, MG

5EDB image
Human Fatty Acid Binding Protein 4 In Complex With 6-Chloro-2-Methyl-4-Phenyl-Quinoline-3-Carboxylic Acid At 1.18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.18 Å Release Date: 2016-03-09
Classification: LIPID BINDING PROTEIN
Ligands: 5M8

5EDC image
Human Fabp4 In Complex With 6-Chloro-4-Phenyl-2-Piperidin-1-Yl-Quinoline-3-Carboxylic Acid At 1.29A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.29 Å Release Date: 2016-03-09
Classification: LIPID BINDING PROTEIN
Ligands: 5M7, SO4

5EDE image
Crystal Structure Of Human Phosphodiesterase 10 In Complex With C13C(Cc(S1)C(Ncc2Occc2)=O)C(Nn3C4Ccc(Cc4)Cl)C, Micromolar Ic50=0.217
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2016-03-09
Classification: HYDROLASE
Ligands: ZN, MG, GOL, 5M6

5EDG image
Crystal Structure Of Human Phosphodiesterase 10 In Complex With C1(C(Nc([Nh]1)Cl)C2Ccccc2)C4=Nn(C3Cccc(C3)Oc(F)(F)F)C=Cc4=O, Micromolar Ic50=0.029618
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2016-03-09
Classification: HYDROLASE
Ligands: ZN, MG, 5MG

5EDH image
Crystal Structure Of Human Phosphodiesterase 10 In Complex With N4C(C)N1C(Nc(N1)Ccc2Nc(Nn2C)N3Cccc3)C(C4)Cc, Micromolar Ic50=0.0037753
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2016-03-09
Classification: HYDROLASE
Ligands: ZN, MG, 5MF

5EDI image
Crystal Structure Of Human Phosphodiesterase 10 In Complex With C2(C(N1Nc(Nc1C(C2)C)Ccc3Nc(Nn3C)N4Cccc4)C)Cl, Micromolar Ic50=0.000279
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2016-03-09
Classification: HYDROLASE
Ligands: ZN, MG, 5M9

5I2R image
Crystal Structure Of Human Phosphodiesterase 10 In Complex With C2(=Nn(C1Cccc(C1)Oc(F)(F)F)C=Cc2=O)C3Ccnn3C4Ccccc4, Micromolar Ic50=0.019462
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2016-03-09
Classification: HYDROLASE
Ligands: ZN, MG, 67A
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