Search Count: 14
![]() |
Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZRU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZRU
![]() |
Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZS3, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZS3, EDO, ACT
![]() |
Crystal Structure Of The Tyk2 Pseudokinase Domain In Complex With Tak-279
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-07-26 Classification: TRANSFERASE Ligands: ZSB, ACT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: ZSB, ACT, EDO
![]() |
Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OVI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OVI
![]() |
Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OVC
![]() |
Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV5
![]() |
Crystal Structure Of Tyk2 Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV0, SO4
![]() |
Crystal Structure Of Jak3 Kinase Domain In Complex With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV5, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV5, CL
![]() |
Crystal Structure Of Jak2 Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2022-08-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: OV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: OV0
![]() |
Escherichia Coli Rna Polymerase In Complex With Squaramide Compound 8.
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:3.57 Å Release Date: 2015-03-11 Classification: transcription/transcription inhibitor Ligands: MG, ZN, 4C6 |
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: MG, ZN, 4C6
![]() |
Escherichia Coli Rna Polymerase In Complex With Squaramide Compound 14 (N-[3,4-Dioxo-2-(4-{[4-(Trifluoromethyl)Benzyl]Amino}Piperidin-1-Yl)Cyclobut-1-En-1-Yl]-3,5-Dimethyl-1,2-Oxazole-4-Sulfonamide)
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:3.82 Å Release Date: 2015-03-11 Classification: transcription/transcription inhibitor Ligands: MG, ZN, 4C2 |
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: MG, ZN, 4C2
![]() |
Escherichia Coli Rna Polymerase In Complex With Myxopyronin B
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:3.84 Å Release Date: 2015-03-11 Classification: transcription/transcription inhibitor Ligands: MG, ZN, 4C4 |
Organism: Escherichia coli o139:h28 (strain e24377a / etec), Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: MG, ZN, 4C4
![]() |
Crystal Structure Of Aminoquinazoline 1 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 242 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 242
![]() |
Crystal Structure Of Aminoquinazoline 36 Bound To Lck
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2007-02-27 Classification: TRANSFERASE Ligands: 1N8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-02-27
Ligands: 1N8
