Search Count: 17
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Crystal Structure Of Tead4 In Complex With Peptide 1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-03-15 Classification: TRANSCRIPTION Ligands: GOL, MYR |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-03-15
Ligands: GOL, MYR
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X-Ray Structure Of Hdm2/Cmr19 At 1.45A: Discovery, X-Ray Structure And Cpp-Conjugation Enabled Uptake Of P53/Mdm2 Macrocyclic Peptide Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-09-22 Classification: LIGASE Ligands: SO4, CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: SO4, CL
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Abl1 In Complex With Compound 7 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: GOL, CL, FYW, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GOL, CL, FYW, STI
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Abl1 In Complex With Compound6 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-12 Classification: TRANSFERASE Ligands: CL, FYH, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: CL, FYH, STI
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Abl1 Kinase (T334I_D382N) In Complex With Asciminib And Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2017-04-05 Classification: TRANSFERASE Ligands: NIL, AY7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-04-05
Ligands: NIL, AY7
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Crystal Structure Of Human Fpps In Complex With Monophosphonate Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2016-07-13 Classification: TRANSFERASE Ligands: 59Z, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: 59Z, PO4
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Crystal Structure Of Human Fpps In Complex With The Monophosphonate Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-07-13 Classification: TRANSFERASE Ligands: 5A7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: 5A7
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Crystal Structure Of Human Fpps In Complex With Biaryl Compound 8E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-10-07 Classification: TRANSFERASE Ligands: 5BL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-07
Ligands: 5BL
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Crystal Structure Of Human Fpps In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 59Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 59Y
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Crystal Structure Of Human Fpps In Complex With Salicylic Acid Derivative 3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: GOL, 5B9, MG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: GOL, 5B9, MG, PO4
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Crystal Structure Of Human Fpps In Complex With Biaryl Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 5BJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 5BJ, PO4
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Crystal Structure Of Human Fpps In Complex With Biaryl Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: GOL, 5BK, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: GOL, 5BK, PO4
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Pak1 In Complex With 2-Chloro-5-Ethyl-8-Fluoro-11-(4-Methylpiperazin-1-Yl)-Dibenzodiazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OQ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OQ, MG
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Pak1 In Complex With (S)-N-(Tert-Butyl)-3-((2-Chloro-5-Ethyl-8-Fluoro-Dibenzodiazepin-11-Yl)Amino)Pyrrolidine-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OR, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OR, MG
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Abl Kinase In Complex With Imatinib And A Fragment (Frag1) In The Myristate Pocket
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: STI, MS9, CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS9, CL
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Abl Kinase In Complex With Imatinib And Fragment (Frag2) In The Myristate Site
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: STI, MS7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS7
