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Search Count: 40

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9GLU image
Crystal Structure Of Krasg12D-Gdp In Complex With The Peptide Mpb1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2025-12-10
Classification: HYDROLASE
Ligands: MG, GDP

9GLW image
Nras-Q61R-Gtp In Complex With The Peptide Mpb2
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2025-12-10
Classification: HYDROLASE
Ligands: MG, GTP

9GLX image
Nras-Q61R-Gtp In Complex With The Peptide Mpb3
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-12-10
Classification: HYDROLASE
Ligands: MG, GTP

9GLZ image
Kras-G12D-Gmppnp In Complex With The Nanobody Km12-Am
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2025-12-10
Classification: HYDROLASE
Ligands: MG, GNP

8C17 image
Crystal Structure Of Tead4 In Complex With Peptide 1
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:2.25 Å Release Date: 2023-03-15
Classification: TRANSCRIPTION
Ligands: GOL, MYR

7KEV image
Pcsk9 In Complex With A Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2021-11-24
Classification: LIPID TRANSPORT, HYDROLASE
Ligands: CA

7KFA image
Pcsk9 In Complex With Pcsk9I A 13Mer Cyclic Peptide Ldlr Disruptor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:2.45 Å Release Date: 2021-11-10
Classification: LIPID TRANSPORT, HYDROLASE
Ligands: CA

7NUS image
X-Ray Structure Of Hdm2/Cmr19 At 1.45A: Discovery, X-Ray Structure And Cpp-Conjugation Enabled Uptake Of P53/Mdm2 Macrocyclic Peptide Inhibitors
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Resolution:1.45 Å Release Date: 2021-09-22
Classification: LIGASE
Ligands: SO4, CL

6R36 image
T. Brucei Farnesyl Pyrophosphate Synthase (Fpps)
Organism: Trypanosoma brucei
Method: X-RAY DIFFRACTION
Resolution:1.67 Å Release Date: 2020-04-08
Classification: TRANSFERASE
Ligands: DMS, PEG

6HD4 image
Abl1 In Complex With Compound 7 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2018-10-24
Classification: TRANSFERASE
Ligands: GOL, CL, FYW, STI

6HD6 image
Abl1 In Complex With Compound6 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2018-09-12
Classification: TRANSFERASE
Ligands: CL, FYH, STI

5MO4 image
Abl1 Kinase (T334I_D382N) In Complex With Asciminib And Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.17 Å Release Date: 2017-04-05
Classification: TRANSFERASE
Ligands: NIL, AY7

5DGM image
Crystal Structure Of Human Fpps In Complex With Monophosphonate Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.86 Å Release Date: 2016-07-13
Classification: TRANSFERASE
Ligands: 59Z, PO4

5DGS image
Crystal Structure Of Human Fpps In Complex With The Monophosphonate Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.62 Å Release Date: 2016-07-13
Classification: TRANSFERASE
Ligands: 5A7

5DJV image
Crystal Structure Of Human Fpps In Complex With Biaryl Compound 8E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2015-10-07
Classification: TRANSFERASE
Ligands: 5BL

5DGN image
Crystal Structure Of Human Fpps In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.08 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 59Y

5DIQ image
Crystal Structure Of Human Fpps In Complex With Salicylic Acid Derivative 3A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: GOL, 5B9, MG, PO4

5DJP image
Crystal Structure Of Human Fpps In Complex With Biaryl Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: 5BJ, PO4

5DJR image
Crystal Structure Of Human Fpps In Complex With Biaryl Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2015-09-30
Classification: TRANSFERASE
Ligands: GOL, 5BK, PO4

4ZLO image
Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2015-08-05
Classification: Transferase/transferase inhibitor
Ligands: 4PV, GOL
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