Search Count: 21
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X-Ray Structure Of Ketohexokinase In Complex With A Pyrimidopyrimidine Analog 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: XNB, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: XNB, SO4
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X-Ray Structure Of Ketohexokinase In Complex With A Pyrimidopyrimidine Analog 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2012-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, XNA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: SO4, XNA
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X-Ray Structure Of Ketohexokinase In Complex With A Pyrimidopyrimidine Analog 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, XNN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-18
Ligands: SO4, XNN
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X-Ray Structure Of Human Chymase In Complex With Small Molecule Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-07-21 Classification: HYDROLASE Ligands: N7O, UNL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-21
Ligands: N7O, UNL
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Cyanofluorophenylacetamides As Orally Efficacious Thrombin Inhibitors
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2009-02-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DKK |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: DKK
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Potent, Nonpeptide Inhibitors Of Human Mast Cell Tryptase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 11M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 11M
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Potent, Nonpeptide Inhibitors Of Human Mast Cell Tryptase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 11N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 11N
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Crystal Structure Of Human Tryptase With Potent Non-Peptide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-02-26 Classification: HYDROLASE Ligands: 2FF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: 2FF
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Glycogen Synthase Kinase-3 Beta In Complex With Bis-(Indole)Maleimide Pyridinophane Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2008-02-19 Classification: TRANSFERASE Ligands: BIM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-19
Ligands: BIM
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X-Ray Structure Of Fxa In Complex With 7-Fluoroindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-01-29 Classification: HYDROLASE Ligands: JNJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-29
Ligands: JNJ
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Discovery Of Potent, Orally Active, Nonpeptide Inhibitors Of Human Mast Cell Chymase By Using Structure-Based Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2007-06-12 Classification: HYDROLASE Ligands: DRX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-06-12
Ligands: DRX
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: NAG, SO4, CO, OHH, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: NAG, SO4, CO, OHH, MES
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A Dual Inhibitor Of The Leukocyte Proteases Cathepsin G And Chymase With Therapeutic Efficacy In Animals Models Of Inflammation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2005-03-01 Classification: HYDROLASE Ligands: SO4, OHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-03-01
Ligands: SO4, OHH
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Potent, Small Molecule Inhibitors Of Human Mast Cell Tryptase. Anti-Asthmatic Action Of A Dipeptide-Based Transition State Analogue Containing Benzothiazole Ketone
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2003-09-23 Classification: HYDROLASE Ligands: CA, SO4, ABB |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-09-23
Ligands: CA, SO4, ABB
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Cathepsin-G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2002-05-01 Classification: HYDROLASE Ligands: KTP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-05-01
Ligands: KTP
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Crystal Structure Of Human Carbonic Anhydrase Ii Complexed With An Anticonvulsant Sugar Sulfamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2002-02-13 Classification: LYASE Ligands: ZN, SMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2002-02-13
Ligands: ZN, SMS
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Crystal Structure Of Human Alpha-Thrombin*Rwj-51438 Complex At 1.7 A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2000-11-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1Z0, NAG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2000-11-03
Ligands: 1Z0, NAG, NA
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Human Thrombin With Active Site N-Methyl-D Phenylalanyl-N-[5-(Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L-Prolinamide Trifluroacetate And Exosite-Hirugen
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1998-05-27 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 00Q, NA |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 1998-05-27
Ligands: 00Q, NA
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Crystal Structures Of Thrombin With Thiazole-Containing Inhibitors: Probes Of The S1' Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1998-04-29 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-04-29
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Thrombin Inhibitor From Theonalla, Cyclotheanamide-Based Macrocyclic Tripeptide Motif
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 1998-03-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 1ZV |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1998-03-18
Ligands: 1ZV