Search Count: 23
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Crystal Structure Of Menin In Complex With Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVE
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Crystal Structure Of Menin In Complex With Inhibitor Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVF, K, EPE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVF, K, EPE, SO4
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Crystal Structure Of Menin In Complex With Inhibitor Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVG
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Inhibitor Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2024-01-03 Classification: HYDROLASE/INHIBITOR Ligands: W8I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: W8I
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Crystal Structure Of Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2024-01-03 Classification: HYDROLASE/INHIBITOR Ligands: WAB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: WAB
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Kras G12D (Gppcp) With Mrtx-1133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2022-03-16 Classification: HYDROLASE/INHIBITOR Ligands: 6IC, GCP, GDP, GOL, ACT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-16
Ligands: 6IC, GCP, GDP, GOL, ACT, MG
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Crystal Structure Of Erk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB, EDO
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Crystal Structure Of Cdk2 In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6QB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 6QB
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Crystal Structure Of Erk2 In Complex With An Inhibitor 14K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-09-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 41B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: 41B
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Discovery Of 5,6,7,8-Tetrahydropyrido[3,4-D]Pyrimidine Inhibitors Of Erk2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-05-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2SH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: 2SH
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Non-Oxime Pyrazole Based Inhibitors Of B-Raf Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2011-05-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: SM7
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Spirocyclic Sulfonamides As Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: SM9
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMH
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Spirochromane Akt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SMR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: SMR
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Human B-Raf Kinase In Complex With A Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FOI
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Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FNI
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Crystal Structure Of Human B-Raf Kinase Domain In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP3
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Crystal Structure Of Human B-Raf Kinase In Complex With A Non-Oxime Furopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-02-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: FP4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-02
Ligands: FP4
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Furo[2,3-C]Pyridine-Based Indanone Oximes As Potent And Selective B-Raf Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2011-01-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SM6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-19
Ligands: SM6
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Discovery Of Dihydrothieno- And Dihydrofuropyrimidines As Potent Pan Akt Inhibitors
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-11-10 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SMY |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-11-10
Ligands: SMY
