Search Count: 31
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Human Pxr Lbd Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 07F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 07F
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Human Pxr Lbd Bound To Gsk003
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 5YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 5YX
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Human Pxr Lbd Bound To Gsk002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 5YU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 5YU
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Human Pxr Lbd Bound To Gsk001
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: P06
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Rip2 Kinase Catalytic Domain Complex With 5Amino1Tertbutyl3(3Methoxyphenyl)1H Pyrazole4Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: M5W, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: M5W, CA
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Rip2 Kinase Catalytic Domain Complex With (5S,6S,8R)-2-(Benzo[D]Thiazol-5-Yl)-6-Hydroxy-4,5,6,7,8,9-Hexahydro-5,8-Methanopyrazolo[1,5-A][1,3]Diazocine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: Q9J, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q9J, CA
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Rip2 Kinase Catalytic Domain Complex With 5-Amino-1-Phenylpyrazole-4-Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2019-10-23 Classification: TRANSFERASE Ligands: M2B, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: M2B, CA
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Rip2 Kinase Catalytic Domain Complex With 2(4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl)Oxy)Ethyl Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: K9T, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: K9T, CA
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Rip2 Kinase Catalytic Domain Complex With 2({4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl}Oxy)Ethan1Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: KA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: KA2
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Crystal Structure Of Rip1 Kinase In Complex With Gsk3145095
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2019-07-03 Classification: TRANSFERASE Ligands: K8K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-03
Ligands: K8K
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Crystal Structure Of Rip1 Kinase In Complex With A Pyrrolidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2019-05-08 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: M5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: M5J, SO4
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Crystal Structure Of Rip1 Kinase In Complex With Dhp77
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: JSW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: JSW
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Amidobenzimidazole (Abzi) Sting Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2018-11-07 Classification: immune system/agonist Ligands: CA, HGJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: CA, HGJ
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Linked Amidobenzimidazole Sting Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-11-07 Classification: immune system/agonist Ligands: HG4, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: HG4, CA
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Rip2 Kinase Catalytic Domain Complex With N(4,5Dimethyl1Hpyrazol3Yl)7Methoxy6(2Methylpropane2Sulfonyl)Quinolin4Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-11-07 Classification: TRANSFERASE Ligands: GEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: GEZ
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Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-07-05 Classification: transferase/transferase inhibitor Ligands: 7MJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: 7MJ
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Compound 3 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GE, SO4
 |
The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Gsk583 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GD
 |
Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 65U
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Rip2 Kinase Catalytic Domain (1 - 310)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2015-10-21 Classification: TRANSFERASE Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-21
Ligands: CA