Search Count: 12
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Cryo-Em Structure Of Cak Modified By Covalent Inhibitor Sy-1365
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-12-25 Classification: TRANSCRIPTION Ligands: A1H46 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-25
Ligands: A1H46
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Cryo-Em Structure Of Cak In Complex With Sy-5609
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-12-25 Classification: TRANSCRIPTION Ligands: YNK |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-12-25
Ligands: YNK
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Cdk2 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2021-11-03 Classification: TRANSFERASE/INHIBITOR Ligands: 3I3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: 3I3
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Structure-Guided Dot1L Probe Optimization By Label-Free Ligand Displacement
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2014-12-03 Classification: Transferase/Transferase inhibitor Ligands: 3US, SO4, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-03
Ligands: 3US, SO4, GOL, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With A Novel Inhibitor Umb32 (N-Tert-Butyl-2-[4-(3,5-Dimethyl-1,2-Oxazol-4-Yl) Phenyl]Imidazo[1,2-A]Pyrazin-3-Amine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2014-10-29 Classification: transcription/transcription inhibitor Ligands: 3P2, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-29
Ligands: 3P2, EDO, GOL
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Epz004777
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: 0QK, SO4, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 0QK, SO4, EDO, UNX
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Crystal Structure Of Human Dot1L In Complex With 2 Molecules Of Epz004777
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: 0QK, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 0QK, UNX
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Sgc0946
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-05-16 Classification: Transferase/Transferase Inhibitor Ligands: BR, AW2, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: BR, AW2, NA
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Sgc0947
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-05-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: AW3, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: AW3, GOL
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Fed2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-05-02 Classification: Transferase/Transferase Inhibitor Ligands: AW0, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
Ligands: AW0, UNX
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Crystal Structure Of Human Dot1L In Complex With Inhibitor Fed1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-05-02 Classification: Transferase/Transferase Inhibitor Ligands: AW1, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
Ligands: AW1, UNX
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Crystal Structure Of Dot1L In Complex With 5-Iodotubercidin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: 5ID, IOD, NA, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: 5ID, IOD, NA, UNX