Search Count: 25
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx3397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P31 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: P31
 |
Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx8512 In The Dfg-In State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: WEG
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx9486 (Bezuclastinib) In The Dfg-In State
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: WEJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: WEJ
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N-Terminal Bromodomain Of Brd4 In Complex With Plx5981
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JC
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 6JE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: 6JE
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N-Terminal Bromodomain Of Brd4 In Complex With Otx-015
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2018-08-01 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: EDO, 6JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: EDO, 6JF
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7904
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 904 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 904
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P06
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx7922
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P02 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: P02
 |
B-Raf Kinase Domain In Complex With Plx5568
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1OO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 1OO, SO4
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx3397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-08-12 Classification: transferase/transferase inhibitor Ligands: P31 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: P31
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Gleevec
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: transferase/transferase inhibitor Ligands: STI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: STI
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Crystal Structure Of Kit Kinase Domain With A Small Molecule Inhibitor, Plx647
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 647 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 647
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Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Plx647-Ome
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-03-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 64M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-27
Ligands: 64M
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B-Raf Kinase V600E Oncogenic Mutant In Complex With Plx4032
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2010-09-22 Classification: transferase/transferase inhibitor Ligands: 032 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-22
Ligands: 032
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Structure Of Ppargamma With 3-(5-Methoxy-1H-Indol-3-Yl)-Propionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-02-17 Classification: TRANSCRIPTION Ligands: ET0, GLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: ET0, GLC
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Structure Of Pparalpha With 3-[5-Methoxy-1-(4-Methoxy-Benzenesulfonyl)-1H-Indol-3-Yl]-Propionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-02-17 Classification: Transcription/Transferase Ligands: ET1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: ET1
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Structure Of Ppardelta With 3-[5-Methoxy-1-(4-Methoxy-Benzenesulfonyl)-1H-Indol-3-Yl]-Propionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2009-02-17 Classification: TRANSCRIPTION Ligands: ET1, 1BO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: ET1, 1BO
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Structure Of Ppargamma With 3-[5-Methoxy-1-(4-Methoxy-Benzenesulfonyl)-1H-Indol-3-Yl]-Propionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2009-02-17 Classification: TRANSCRIPTION Ligands: ET1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: ET1
 |
B-Raf Kinase In Complex With Plx4720
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2008-02-26 Classification: TRANSFERASE Ligands: 324 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: 324