Search Count: 27
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Structure Of 1 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1P
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Structure Of 5 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1R
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Structure Of 10 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, WYU
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Structure Of 12 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1Z
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Structure Of 18 (Bi-2493) In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, VU6
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Crystal Structure Of The Brd9 Bromodomain With Bi-7189
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-06-21 Classification: GENE REGULATION Ligands: M2O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: M2O
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Kras-G12V In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.02 Å Release Date: 2023-06-21 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: GDP, MG, EDO, OFU
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Kras In Complex With Precursor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, LR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, LR4
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Kras In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
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Kras-G12C In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
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Kras-G12D In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
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Kras-G13D In Complex With Bi-2865
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2023-06-07 Classification: ONCOPROTEIN Ligands: GDP, MG, EDO, OFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, OFU
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Kras-G13D In Complex With Bi-2493
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2023-06-07 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: GDP, MG, EDO, VU6
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Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
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Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
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Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
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Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
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Crystal Structure Of The Bptf Bromodomain In Complex With Bi-7190
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.03 Å Release Date: 2022-08-31 Classification: PROTEIN BINDING Ligands: M1I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: M1I
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Crystal Structure Of Crystal Form 2 Of An Active Kras G12D (Gppcp) Dimer In Complex With Bi-5747
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-11-18 Classification: SIGNALING PROTEIN Ligands: MG, GCP, R6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: MG, GCP, R6W
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: GCP, MG, F0N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GCP, MG, F0N
