Search Count: 17
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Crystal Structure Of Brd4-Bd1 In Complex With Nvs-Bet-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2020-12-23 Classification: TRANSCRIPTION Ligands: QFN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: QFN
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Human Malt1(329-729) In Complex With A Chromane Urea Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-12-09 Classification: HYDROLASE Ligands: RJK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: RJK
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Human Malt1(329-729) In Complex With A Chromane Urea Containing Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2020-12-09 Classification: HYDROLASE Ligands: RJH, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: RJH, MG
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Abl1 In Complex With Compound 7 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: GOL, CL, FYW, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GOL, CL, FYW, STI
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Abl1 In Complex With Compound6 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-12 Classification: TRANSFERASE Ligands: CL, FYH, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: CL, FYH, STI
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Human Vascular Endothelial Growth Factor Receptor 2 (Kdr) Kinase Domain In Complex With Aal993
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-12-16 Classification: TRANSFERASE Ligands: 5T2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 5T2
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Structural Basis Of Jak2 Inhibition By The Type Ii Inhibtor Nvp-Bbt594
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2012-05-16 Classification: Transferase/transferase inhibitor Ligands: 046, MLI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: 046, MLI
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Discovery Of A Small Molecule Type Ii Inhibitor Of Wild-Type And Gatekeeper Mutants Of Bcr-Abl, Pdgfralpha, Kit, And Src Kinases
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-02-15 Classification: TRANSFERASE Ligands: NG7, MES, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-02-15
Ligands: NG7, MES, GOL
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Structure Of Abl Kinase In Complex With Imatinib And Gnf-2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: STJ, STI, CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: STJ, STI, CL
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Human Abl Kinase In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: NIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NIL
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Human Abl Kinase Domain In Complex With Imatinib (Sti571, Glivec)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: STI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: STI
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Abl Kinase Domain In Complex With Nvp-Aeg082
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: GIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: GIN
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Abl Kinase Domain Unligated And In Complex With Tetrahydrostaurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: 4ST |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: 4ST
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Abl Kinase Domain In Complex With Pd180970
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: JIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: JIN
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Abl Kinase Domain In Complex With Nvp-Afg210
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: KIN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: KIN
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Structure Of Unphosphorylated C-Src In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2005-06-21 Classification: TRANSFERASE Ligands: SO4, MPZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-21
Ligands: SO4, MPZ
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Crystal Structure Of The Jak3 Kinase Domain In Complex With A Staurosporine Analogue
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2005-05-24 Classification: TRANSFERASE Ligands: DTV, 4ST |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-05-24
Ligands: DTV, 4ST
