Search Count: 47
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Crystal Structure Of Cdk2 In Complex With Cyclin A Inhibitor 6-[(E)-2-(4-Chlorophenyl)Ethenyl]-2-{[(2R)-3-(4-Hydroxyphenyl)-1-Methoxy-1-Oxopropan-2-Yl]Carbamoyl}Quinoline-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: OW6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: OW6
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Atp-Competitive Partial Antagonists-'Pair'S-Rheostatically Modulate Ire1Alpha'S Kinase Helix-Alphac To Segregate Its Rnase-Mediated Biological Outputs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-29 Classification: UNKNOWN FUNCTION Ligands: U4N, GOL, EDO, PEG, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: U4N, GOL, EDO, PEG, PGE
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C-Src Bound To Atp-Competitive Inhibitor I14
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-06-17 Classification: TRANSFERASE/INHIBITOR Ligands: I14 |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: I14
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Crystal Structure Of The Designed Protein Dncr2/Danoprevir/Ns3A Complex
Organism: Hepacivirus c, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2019-09-11 Classification: DE NOVO PROTEIN/HYDROLASE/INHIBITOR Ligands: ZN, TSV, SO4 |
Organism: Hepacivirus c, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: ZN, TSV, SO4
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Calcium-Dependent Protein Kinase 1 From Toxoplasma Gondii (Tgcdpk1) In Complex With Inhibitor Uw1553
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-12-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: UW5 |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2017-12-06
Ligands: UW5
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C-Src V281C Kinase Domain In Complex With Rao-Iv-156
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2017-09-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: S56 |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: S56
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C-Src Kinase Domain In Complex With Rao-Iv-151
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-08-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 73A |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: 73A
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C-Src V281C Kinase Domain In Complex With Rao-Iv-151
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-08-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 71D |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 71D
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C-Src V281C Bound To N-[3-({6-[(1E)-2-Cyano-3-(Methylamino)-3-Oxoprop-1-En-1-Yl]-7-(2-Methoxyethyl)-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Ethynyl)-4-Methylphenyl]-3-(Trifluoromethyl)Benzamide Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-08-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 72F |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 72F
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Crystal Structure Of Apo Human Ire1 Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2016-06-08 Classification: Transferase/Oxidoreductase Ligands: CS, NA, GOL, DTT, BME, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: CS, NA, GOL, DTT, BME, CL
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Src Kinase In Complex With A Sulfonamide Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-06-01 Classification: Transferase/Transferase Inhibitor Ligands: 6G3 |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2016-06-01
Ligands: 6G3
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Calcium-Dependent Protein Kinase From Eimeria Tenella In Complex With Adp
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: CA, MG, ADP |
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: CA, MG, ADP
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Calcium-Dependent Protein Kinase From Eimeria Tenella
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: CA |
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: CA
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Cdpk1 From Eimeria Tenella In Complex With Inhibitor Uw1354
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-04-06 Classification: Transferase/Transferase Inhibitor Ligands: CA, KS1 |
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: CA, KS1
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Cdpk1 From Eimeria Tenella In Complex With Inhibitor Uw1521
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-04-06 Classification: Transferase/Transferase Inhibitor Ligands: CA, BK8 |
Organism: Eimeria tenella
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: CA, BK8
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Calcium-Dependent Protein Kinase 1 From Toxoplasma Gondii (Tgcdpk1) In Complex With Inhibitor Uw1647
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-10-15 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: UW3 |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: UW3
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Calcium-Dependent Protein Kinase 1 From Toxoplasma Gondii (Tgcdpk1) In Complex With Inhibitor Uw1561
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-08-27 Classification: TRANSFERASE Ligands: UW2 |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2014-08-27
Ligands: UW2
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A Double Mutant Rat Erk2 In Complex With A Pyrazolo[3,4-D]Pyrimidine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2H1 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-04-16
Ligands: 2H1
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Calcium-Dependent Protein Kinase 1 From Toxoplasma Gondii (Tgcdpk1) In Complex With Inhibitor Uw1268
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2014-03-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: V68 |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: V68
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Calcium-Dependent Protein Kinase 1 From Toxoplasma Gondii (Tgcdpk1) In Complex With Inhibitor Uw1517
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-03-19 Classification: Transferase/Transferase Inhibitor Ligands: UW1 |
Organism: Toxoplasma gondii
Method: X-RAY DIFFRACTION
Release Date: 2014-03-19
Ligands: UW1
