Search Count: 17
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Brafv600E Kinase Domain In Complex With Chemically Linked Vemurafenib Inhibitor Vem-6-Vem
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2016-09-14 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6N9, DMS, GOL, TMA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6N9, DMS, GOL, TMA
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Brafv600E Kinase Domain In Complex With Chemically Linked Vemurafenib Inhibitor Vem-3-Vem
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2016-09-14 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: DMS, BEN, EOH, 6NB, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: DMS, BEN, EOH, 6NB, CL, GOL
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Brafv600E Kinase Domain In Complex With Chemically Linked Vemurafenib Inhibitor Vem-Bisamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-09-14 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: BEN, 6NC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: BEN, 6NC
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound G-5555
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59T
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Crystal Structure Of Pak1 In Complex With An Inhibitor Compound Frax1036
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-01-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 59U, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 59U, DMS
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Crystal Structure Of P300 Histone Acetyltransferase Domain In Complex With Coenzyme A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2014-06-11 Classification: TRANSFERASE Ligands: PEG, DMS, COA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: PEG, DMS, COA
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Crystal Structure Of P300 Histone Acetyltransferase Domain In Complex With Acetyl-Coenzyme A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2014-06-11 Classification: TRANSFERASE Ligands: ACO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: ACO, DMS
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Crystal Structure Of P300 Histone Acetyltransferase Domain In Complex With An Inhibitor, Acetonyl-Coenzyme A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SOP, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: SOP, DMS
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Crystal Structure Of Pak1 Kinase Domain In Complex With Frax597 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2013-08-28 Classification: transferase/transferase inhibitor Ligands: XR1, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: XR1, CL
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Crystal Structure Of Pak1 Kinase Domain With The Ruthenium Phthalimide Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0H2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: 0H2
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Structure Of Death-Associated Protein Kinase 1 (Dapk1) In Complex With A Ruthenium Octasporine Ligand (Osv)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-04-27 Classification: TRANSFERASE Ligands: OSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-27
Ligands: OSV
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Structure Of Glycogen Synthase Kinase 3 Beta (Gsk3B) In Complex With A Ruthenium Octasporine Ligand (Os1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2010-12-22 Classification: TRANSFERASE Ligands: OS1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: OS1
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Crystal Structure Of Pak1 Kinase Domain With Ruthenium Complex Dw1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2009-03-03 Classification: TRANSFERASE Ligands: DW1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-03
Ligands: DW1
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Crystal Structure Of Pak1 Kinase Domain With Ruthenium Complex Lambda-Fl172
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2009-02-17 Classification: TRANSFERASE Ligands: FLL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: FLL
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Extremely Tight Binding Of Ruthenium Complex To Glycogen Synthase Kinase 3
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2008-12-09 Classification: TRANSFERASE Ligands: AG1 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: AG1
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Crystal Structure Of The Human Pim1 In Complex With An Osmium Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2008-06-24 Classification: TRANSFERASE Ligands: SO4, DWC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-24
Ligands: SO4, DWC
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Crystal Structure Of Human Pim1 In Complex With Fluorinated Ruthenium Pyridocarbazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-04-10 Classification: TRANSFERASE Ligands: CL, JM1, EDO, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-04-10
Ligands: CL, JM1, EDO, EPE
