Search Count: 27
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Crystal Structure Of The Pwwp1 Domain Of Nsd2 Bound By Compound 11.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: A1IFS, A1IEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1IFS, A1IEG
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Crystal Structure Of The Pwwp1 Domain Of Nsd2 Bound By Compound 7.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: A1IEF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1IEF
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of The P110Alpha Catalytic Subunit From Homo Sapiens In Complex With Activator 1938
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2023-05-24 Classification: TRANSFERASE Ligands: QIH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: QIH
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Crystal Structure Of The Apo P110Alpha Catalytic Subunit From Homo Sapiens
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2023-02-15 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
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Crystal Structure Of Wild-Type C-Met Bound By Compound 7.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2022-08-31 Classification: TRANSFERASE Ligands: SO4, MDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: SO4, MDI
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Crystal Structure Of D1228V C-Met Bound By Compound 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-08-31 Classification: TRANSFERASE Ligands: GOL, MDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: GOL, MDI
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Crystal Structure Of Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-08-24 Classification: TRANSFERASE Ligands: PO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: PO4, GOL
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Crystal Structure Of Pi3Kalpha In Complex With The Inhibitor Nvp-Byl719
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-08-24 Classification: TRANSFERASE Ligands: 1LT, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 1LT, NA
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Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2YE
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Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F97, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: F97, EDO, MES
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Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2WI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2WI, SO4
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Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2TR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2TR
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Structure Of Mature Activin A With Small Molecule 42
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-02-03 Classification: SIGNALING PROTEIN Ligands: SO4, OCK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-03
Ligands: SO4, OCK
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Structure Of Mature Activin A With Small Molecule 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2021-01-13 Classification: SIGNALING PROTEIN Ligands: ODQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: ODQ, SO4
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Pandda Analysis Group Deposition -- Crystal Structure Of Human Cleavage Factor Im In Complex With Nm450-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2020-07-08 Classification: RNA BINDING PROTEIN Ligands: ZN, ACT, RVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-08
Ligands: ZN, ACT, RVY
