Search Count: 16
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Pi3Kg In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: DD8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: DD8
 |
Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: GQD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: GQD
 |
Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 2.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: QHG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: QHG
 |
Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: J0W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: J0W
 |
Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 4.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: 7QN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 7QN
 |
Selective Estrogen Receptor Downregulator Antagonists: Tetrahydroisoquinoline Phenols 5.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2016-02-10 Classification: SIGNALING PROTEIN Ligands: VQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: VQI
 |
A Novel Oral Selective Estrogen Receptor Down-Regulator, Azd9496, Drives Tumour Growth Inhibition In Estrogen Receptor Positive And Esr1 Mutant Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2015-12-16 Classification: SIGNALING PROTEIN Ligands: KE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: KE9
 |
Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: XBR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: XBR
 |
Optimization Of A Novel Binding Motif To To (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-Fluoro-2-Methylpropyl)-3-Methyl-2,3,4,9-Tetrahydro-1H- Pyrido(3,4-B)Indol-1-Yl)Phenyl)Acrylic Acid (Azd9496), A Potent And Orally Bioavailable Selective Estrogen Receptor Downregulator And Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-10-14 Classification: SIGNALING PROTEIN Ligands: GW5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: GW5
 |
Oxyphenylpropenoic Acids As Oral Selective Estrogen Receptor Down- Regulators.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2015-04-22 Classification: SIGNALING PROTEIN Ligands: 85Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: 85Z
 |
Cathepsin K Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-07-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0LB, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0LB, GOL
 |
Cathepsin K Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2012-07-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0LC, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0LC, SO4, GOL
 |
Mmp13 In Complex With A Novel Selective Non Zinc Binding Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-06-29 Classification: HYDROLASE Ligands: 5EL, ZN, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-29
Ligands: 5EL, ZN, CA, NA
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Human Serum Albumin In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IMX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: IMX
 |
Human Serum Albumin In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IPX, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: IPX, PO4
 |
Human Serum Albumin In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-10-27 Classification: TRANSPORT PROTEIN Ligands: IQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: IQX