Search Count: 39
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Structure Of Bovine Pka Bound To (R)-N-(4-(1H-Pyrrolo[2,3-B]Pyridin-4-Yl)Phenyl)-2-Amino-4-Methylpentanamide
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-02-21 Classification: CYTOSOLIC PROTEIN Ligands: ZWG |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: ZWG
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Sars-Cov-2 3Clpro In Complex With N-(4-(1H-Pyrazol-4-Yl)Phenyl)-N-(3-Chlorobenzyl)-2-(Pyridin-3-Yl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-01-11 Classification: VIRAL PROTEIN,HYDROLASE/INHIBITOR Ligands: I2D |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2023-01-11
Ligands: I2D
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Sars-Cov-2 3Clpro In Complex With N-(4-(1H-Imidazol-4-Yl)Phenyl)-N-(3-Chloro-5-Fluorobenzyl)-2-(Isoquinolin-4-Yl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-01-11 Classification: VIRAL PROTEIN,HYDROLASE/INHIBITOR Ligands: I2N |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2023-01-11
Ligands: I2N
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Sars-Cov-2 3Clpro In Complex With 2-(Benzotriazol-1-Yl)-N-[4-(1H-Pyrazol-4-Yl)Phenyl]-N-(3-Thienylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, hydrolase/Inhibitor Ligands: Y6A |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6A
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Sars-Cov-2 3Clpro In Complex With N-[4-[[2-(Benzotriazol-1-Yl)Acetyl]-(3-Thienylmethyl)Amino]Phenyl]Cyclopropanecarboxamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6J |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6J
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Sars-Cov-2 3Clpro In Complex With 2-(Benzotriazol-1-Yl)-N-[4-(1H-Imidazol-4-Yl)Phenyl]-N-(3-Thienylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6G |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6G
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Sars-Cov-1 3Clpro In Complex With N-(4-(1H-Imidazol-4-Yl)Phenyl)-2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(Thiophen-3-Ylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: GOL, Y6G, PEG |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: GOL, Y6G, PEG
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Sars-Cov-1 3Clpro In Complex With 2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(4-(Pyridin-3-Yl)Phenyl)-N-(Thiophen-3-Ylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: Y6D, GOL |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: Y6D, GOL
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Sars-Cov-1 3Clpro In Complex With N-(4-(1H-Pyrazol-4-Yl)Phenyl)-2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(Thiophen-3-Ylmethyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: GOL, Y6A |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: GOL, Y6A
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Sars-Cov-1 3Clpro In Complex With 2-(1H-Benzo[D][1,2,3]Triazol-1-Yl)-N-(3-Chlorobenzyl)-N-(4-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl)Acetamide
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-08-11 Classification: VIRAL PROTEIN, Hydrolase/Inhibitor Ligands: PEG, GOL, Y67 |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: PEG, GOL, Y67
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Wdr5 In Complex With Myc Site Fragment Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: Q8G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: Q8G
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Wdr5 In Complex With Myc Site Fragment Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: Q8D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: Q8D
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonmides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: Q8P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: Q8P
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonmides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: Q8M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: Q8M
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonmides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: Q8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: Q8S
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonamides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: QBS, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: QBS, SO4, DMS
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonamides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: QBP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: QBP
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonamides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: QBM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: QBM
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Discovery Of Fragment-Inspired Heterocyclic Benzenesulfonmides As Inhibitors Of The Wdr5-Myc Interaction
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2020-04-15 Classification: TRANSCRIPTION Ligands: QF1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-15
Ligands: QF1
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Discovery And Structure-Based Optimization Of Potent And Selective Wdr5 Inhibitors Containing A Dihydroisoquinolinone Bicyclic Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-01-01 Classification: TRANSCRIPTION Ligands: Q41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-01
Ligands: Q41
