Search Count: 16
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Discovery Of A Small Molecule Itk And Pan-Trk Kinase Inhibitor (Pf-07245303) For The Potential Topical Treatment Of Atopic Dermatitis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-11-19 Classification: SIGNALING PROTEIN Ligands: A1B66 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-19
Ligands: A1B66
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Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG4
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Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG5
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Design And Application Of Synthetic 17B-Hsd13 Substrates To Drug Discovery, And To Reveal Preserved Catalytic Activity Of Protective Human Variants
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: NAD, A1AG6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: NAD, A1AG6
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Crystal Structures Of Hsd17B13 Complexes
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2023-08-09 Classification: OXIDOREDUCTASE Ligands: NAD |
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION
Release Date: 2023-08-09
Ligands: NAD
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Hsd17B13 In Complex With Cofactor And Inhibitor
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2023-08-09 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NAD, YXW |
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION
Release Date: 2023-08-09
Ligands: NAD, YXW
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Crystal Structures Of 17-Beta-Hydroxysteroid Dehydrogenase 13
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2023-08-09 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NAD, YXW |
Organism: Canis lupus familiaris
Method: X-RAY DIFFRACTION
Release Date: 2023-08-09
Ligands: NAD, YXW
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Crystal Structures Of 17-Beta-Hydroxysteroid Dehydrogenase 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2023-08-09 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NAD, YYC, CE1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-09
Ligands: NAD, YYC, CE1, SO4
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Cryo-Em Structure Of Human Ace2 Receptor Bound To Protein Encoded By Vaccine Candidate Bnt162B1
Organism: Homo sapiens, Severe acute respiratory syndrome coronavirus 2, Human immunodeficiency virus 1
Method: ELECTRON MICROSCOPY Release Date: 2021-02-24 Classification: VIRAL PROTEIN |
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Cryo-Em Structure Of Protein Encoded By Vaccine Candidate Bnt162B2
Organism: Severe acute respiratory syndrome coronavirus 2
Method: ELECTRON MICROSCOPY Release Date: 2021-02-24 Classification: VIRAL PROTEIN |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: ELECTRON MICROSCOPY
Release Date: 2021-02-24
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Crystal Structure Of A Human Lysosome Resident Glycoprotein, Lysosomal Acid Lipase, And Its Implications In Cholesteryl Ester Storage Disease (Cesd)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2020-06-17 Classification: HYDROLASE Ligands: NAG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: NAG, SO4
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Crystal Structure Of T Brucei Phosphodiesterase B2 Bound To Compound 13E
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2017-11-01 Classification: HYDROLASE Ligands: ZN, MG, LLI |
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ZN, MG, LLI
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Crystal Structure Of T Brucei Phosphodiesterase B2 Bound To Compound 15B
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-11-01 Classification: HYDROLASE Ligands: ZN, MG, LLN |
Organism: Trypanosoma brucei brucei
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: ZN, MG, LLN
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Mycobacterium Tuberculosis Inha Bound To Nitd-564
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-01-21 Classification: OXIDOREDUCTASE Ligands: NAD, 3KX |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2015-01-21
Ligands: NAD, 3KX
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Mycobacterium Tuberculosis Inha Bound To Nitd-916
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2015-01-21 Classification: OXIDOREDUCTASE Ligands: NAD, 3KY |
Organism: Mycobacterium tuberculosis h37rv
Method: X-RAY DIFFRACTION
Release Date: 2015-01-21
Ligands: NAD, 3KY
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Quadruple Mutant(N51I+C59R+S108N+I164L) Plasmodium Falciparum Dihydrofolate Reductase-Thymidylate Synthase(Pfdhfr-Ts) Complexed With Qn254, Nadph, And Dump
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-07-28 Classification: OXIDOREDUCTASE, TRANSFERASE Ligands: KA5, NDP, UMP |
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: KA5, NDP, UMP
