Search Count: 17
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAH, LUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAH, LUP
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, EDO, SAM, L0J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, EDO, SAM, L0J
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, SAM, O41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, SAM, O41
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Co-Crystal Structure Of Human Smyd3 With Isoxazole Amides Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2020-01-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, MG, GOL, SAM, O6A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: ZN, MG, GOL, SAM, O6A
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Discovery Of Potent And Selective Covalent Protein Arginine Methyltransferase (Prmt5) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-06-19 Classification: TRANSFERASE Ligands: CUX, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-19
Ligands: CUX, DMS, EDO
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Crystal Structure Of Human Hexokinase 2 With Cmpd 30, A 2-Amino-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 604 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 604
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Crystal Structure Of Human Hexokinase 2 With Cmpd 27, A 2-Amido-6-Benzenesulfonamide Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 603 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 603
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Crystal Structure Of Human Hexokinase 2 With Cmpd 1, A C-2-Substituted Glucosamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2016-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 62C, BG6, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-30
Ligands: 62C, BG6, FLC
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Structure Of Pka With A Protein Kinase B-Selective Inhibitor.
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-12-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B99 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: B99
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Structure Of Pi3K Gamma With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-06-30 Classification: TRANSFERASE Ligands: SO4, LXX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-30
Ligands: SO4, LXX
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Structure Of Pi3K Gamma With A Potent Inhibitor: Gsk2126458
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-06-23 Classification: TRANSFERASE Ligands: SO4, ZIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-23
Ligands: SO4, ZIG
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SB3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SB3
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SBX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SBX
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Design, Synthesis, And Kinetic Evaluation Of High-Affinity Fkbp Ligands, And The X-Ray Crystal Structures Of Their Complexes With Fkbp12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1994-01-31 Classification: CIS-TRANS ISOMERASE Ligands: SB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 1994-01-31
Ligands: SB1
