Search Count: 25
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Structure Of Bfl1 In Complex With A Covalent Inhibitor, Alternative Series, Cmpd25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2026-01-14 Classification: APOPTOSIS Ligands: A1JL2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-14
Ligands: A1JL2
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Structure Of Chip E3 Ubiquitin Ligase Tpr Domain In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-08-27 Classification: LIGASE Ligands: A1I6K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1I6K, SO4
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Structure Of Chip E3 Ubiquitin Ligase Tpr Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2025-08-27 Classification: LIGASE Ligands: A1I5T, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1I5T, SO4
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Structure Of Chip E3 Ubiquitin Ligase Tpr Domain In Complex With Compound 8.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2025-08-27 Classification: LIGASE Ligands: A1I6J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1I6J, EDO
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Structure Of Chip E3 Ubiquitin Ligase Tpr Domain In Complex With Compound 9.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2025-08-27 Classification: LIGASE Ligands: A1I6I, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1I6I, SO4
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Fragment Screening Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2025-06-18 Classification: GENE REGULATION Ligands: A1I5P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1I5P, ZN
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Tricyclic Pyrimidoindolone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-05-14 Classification: GENE REGULATION Ligands: A1I45, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1I45, ZN
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Crystal Structure Of The Vhl-Eloc-Elob Complex With A Covalent Compound Bound To C77 Of Vhl.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2025-03-26 Classification: LIGASE Ligands: 3JF, A1IMD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: 3JF, A1IMD
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Bfl1 Covalently Bound To Inhibitor Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-12-18 Classification: APOPTOSIS Ligands: A1ILY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1ILY
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Bfl1 Covalently Bound To Inhibitor Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-12-18 Classification: APOPTOSIS Ligands: BUD, A1ILV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: BUD, A1ILV
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Bfl1 Covalently Bound To Inhibitor Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.08 Å Release Date: 2024-12-18 Classification: APOPTOSIS Ligands: A1ILX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1ILX
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Bfl1 Covalently Bound To Inhibitor Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2024-12-18 Classification: APOPTOSIS Ligands: A1ILU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1ILU
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Bfl1 Covalently Bound To Inhibitor Compound 43
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.15 Å Release Date: 2024-12-18 Classification: APOPTOSIS Ligands: A1ILW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1ILW
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDP
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDO
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Discovery Of A Series Of Covalent, Cell Active Bfl-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2024-10-02 Classification: APOPTOSIS Ligands: A1IDG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: A1IDG
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Bfl1 In Complex With A Reversible Covalent Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2024-07-03 Classification: APOPTOSIS Ligands: A1H2C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: A1H2C
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Structure Of The Human Ddb1-Dda1-Dcaf15 E3 Ubiquitin Ligase Bound To Compound Furan 12
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-03 Classification: LIGASE Ligands: A1H17 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-03
Ligands: A1H17
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Structure Of The Human Ddb1-Dda1-Dcaf15 E3 Ubiquitin Ligase Bound To Compound Furan 24
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-04-03 Classification: LIGASE Ligands: A1H18 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-04-03
Ligands: A1H18
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C-Terminal Bromodomain Of Human Brd2 With N5-((1R,5S,6R)-3-Oxabicyclo[3.1.0]Hexan-6-Yl)-3-(1H-Indol-4-Yl)-N7-Methyl-2,3-Dihydrobenzofuran-5,7-Dicarboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2021-07-28 Classification: NUCLEAR PROTEIN Ligands: EDO, V9Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: EDO, V9Q
