Search Count: 18
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Nicotinamide Riboside And Cd38: Covalent Inhibition And Live-Cell Labeling
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-11-06 Classification: HYDROLASE/INHIBITOR Ligands: NNR, RIB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: NNR, RIB
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X-Ray Structure Of Human Cd38 Catalytic Domain With 2'-Cl-Aranad+
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-06-03 Classification: HYDROLASE Ligands: ROJ, K, PO4, PEG, MPD, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: ROJ, K, PO4, PEG, MPD, PGE
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Development Of Alkyl Glycerone Phosphate Synthase Inhibitors: Complex With Inhibitor 2I
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-01-02 Classification: FLAVOPROTEIN Ligands: FAD, F6T |
Organism: Cavia porcellus
Method: X-RAY DIFFRACTION
Release Date: 2019-01-02
Ligands: FAD, F6T
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Crystal Structure Of Human Cd38 In Complex With 4'-Thioribose Nad+
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-11-21 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZNA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: ZNA
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Crystal Structure Of Pde10A With A Biaryl Ether Inhibitor ((1-(3-(4-((1H-Benzo[D]Imidazol-2-Yl)Amino)Phenoxy)Pyridin-2-Yl)Piperidin-4-Yl)Methanol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-12-12 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, SO4, 15J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-12
Ligands: ZN, SO4, 15J
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Crystal Structure Of Pde10A With A Biaryl Ether Inhibitor (1-(1-(3-(4-(Benzo[D]Thiazol-2-Ylamino)Phenoxy)Pyrazin-2-Yl)Piperidin-4-Yl)Ethanol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-12-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, GOL, 15H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-12
Ligands: ZN, SO4, GOL, 15H
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Crystal Structure Of Bace1 In Complex With Hydroxyethylamine Inhibitor 37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0K9, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: 0K9, GOL
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Crystal Structure Of Bace1 In Complex With Biarylspiro Aminooxazoline 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2012-09-12 Classification: HYDROLASE/INHIBITOR Ligands: IOD, DWA, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-12
Ligands: IOD, DWA, DMS
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Crystal Structure Of Bace1 In Complex With Aminooxazoline Xanthene 9L
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2012-09-12 Classification: HYDROLASE/INHIBITOR Ligands: IOD, DWB, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-12
Ligands: IOD, DWB, GOL, DMS
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Crystal Structure Of Bace1 In Complex With Aminooxazoline Xanthene 11A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-09-12 Classification: HYDROLASE/INHIBITOR Ligands: IOD, DWD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-12
Ligands: IOD, DWD, GOL
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Structure Of Bace-1 (Beta-Secretase) In Complex With (2R)-N-((2S,3R)-1-(Benzo[D][1,3]Dioxol-5-Yl)-3-Hydroxy-4-((S)-6'-Neopentyl-3',4'-Dihydrospiro[Cyclobutane-1,2'-Pyrano[2,3-B]Pyridine]-4'-Ylamino)Butan-2-Yl)-2-Methoxypropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-04-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: IOD, GOL, 0KN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-18
Ligands: IOD, GOL, 0KN
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Structure Of Bace-1 (Beta-Secretase) In Complex With (R)-3-(2-Amino-6-O-Tolylquinolin-3-Yl)-N-((R)-2,2-Dimethyltetrahydro-2H-Pyran-4-Yl)-2-Methylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, 3RS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, 3RS
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Structure Of Bace-1 (Beta-Secretase) In Complex With 6-(Thiophen-3-Yl)Quinolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, RSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, RSV
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Structure Of Bace-1 (Beta-Secretase) In Complex With 6-(2-(3,3-Dimethylbut-1-Ynyl)Phenyl)Quinolin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, RTH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, RTH
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Aminoquinolin-3-Yl)-N-Cyclohexyl-N-Methylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RTM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RTM
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Amino-6-O-Tolylquinolin-3-Yl)-N-Cyclohexylpropanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RTN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RTN
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Structure Of Bace-1 (Beta-Secretase) In Complex With 3-(2-Aminoquinolin-3-Yl)-N-(Cyclohexylmethyl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, 3RU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, 3RU
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Structure Of Bace-1 (Beta-Secretase) In Complex With 2-((2-Amino-6-O-Tolylquinolin-3-Yl)Methyl)-N-(Cyclohexylmethyl)Pentanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2011-08-31 Classification: Hydrolase/Hydrolase Inhibitor Ligands: IOD, GOL, RVI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: IOD, GOL, RVI
