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4I0D image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4I1F image
Structure Of Parkin-S223P E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.58 Å Release Date: 2013-06-19
Classification: LIGASE
Ligands: ZN, BA

4I1H image
Structure Of Parkin E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2013-06-19
Classification: LIGASE
Ligands: ZN

4HZT image
Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates

4I0E image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4I0F image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4I0G image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4I0Z image
Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates

4I10 image
Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates

4I11 image
Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates.

4I12 image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4I1C image
Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors

4AN2 image
Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2012-12-19
Classification: TRANSFERASE
Ligands: EUI, ACP, MG

4AN3 image
Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.10 Å Release Date: 2012-12-19
Classification: TRANSFERASE
Ligands: MG, ATP, 5Y0

4AN9 image
Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.80 Å Release Date: 2012-12-19
Classification: TRANSFERASE
Ligands: ACP, MG, 2P7

4ANB image
Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2012-12-19
Classification: TRANSFERASE
Ligands: YQY, ACP, MG

4AWO image
Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2012-08-29
Classification: CHAPERONE
Ligands: 99B

4AWP image
Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.82 Å Release Date: 2012-08-29
Classification: CHAPERONE
Ligands: 99A

4AWQ image
Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2012-08-29
Classification: CHAPERONE
Ligands: 592

4ANU image
Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.81 Å Release Date: 2012-05-09
Classification: TRANSFERASE
Ligands: SO4, EM7
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