Search Count: 34
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-10-09 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: ZN, 1B7
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Structure Of Parkin-S223P E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2013-06-19 Classification: LIGASE Ligands: ZN, BA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: ZN, BA
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Structure Of Parkin E3 Ligase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-06-19 Classification: LIGASE Ligands: ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-19
Ligands: ZN
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 0ZA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 0ZA
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B8
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BF
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1B9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1B9
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: 1BB, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BB, ZN
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BS
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Structure-Based Design Of Novel Dihydroisoquinoline Bace-1 Inhibitors That Do Not Engage The Catalytic Aspartates.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2013-03-06 Classification: transferase/transferase inhibitor Ligands: ZN, 1CH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1CH
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: 1BC, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: 1BC, ZN, NA
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Design And Synthesis Of Thiophene Dihydroisoquinolins As Novel Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-03-06 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 1BE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: ZN, 1BE
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: EUI, ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: EUI, ACP, MG
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: MG, ATP, 5Y0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: MG, ATP, 5Y0
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: ACP, MG, 2P7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: ACP, MG, 2P7
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Crystal Structures Of Human Mek1 With Carboxamide-Based Allosteric Inhibitor Xl518 (Gdc-0973), Or Related Analogs.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-12-19 Classification: TRANSFERASE Ligands: YQY, ACP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: YQY, ACP, MG
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 99B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 99B
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 99A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 99A
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Complex Of Hsp90 Atpase Domain With Tropane Derived Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-08-29 Classification: CHAPERONE Ligands: 592 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 592
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Complexes Of Pi3Kgamma With Isoform Selective Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2012-05-09 Classification: TRANSFERASE Ligands: SO4, EM7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-09
Ligands: SO4, EM7
