Search Count: 10
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Structure Of Kras G12C Bound To Inhibitor 13Ab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-04-15 Classification: ONCOPROTEIN Ligands: CA, A1C6Y, GOL, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-15
Ligands: CA, A1C6Y, GOL, GDP
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Structure Of Kras G12C Bound To Inhibitor 13Ba
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2026-04-15 Classification: ONCOPROTEIN Ligands: GDP, A1C60, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-15
Ligands: GDP, A1C60, CA
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[Fefe]-Hydrogenase From D. Desulfuricans With Synthetic Active Site Containing Only One Cyanide Ligand.
Organism: Desulfovibrio desulfuricans
Method: X-RAY DIFFRACTION Resolution:0.96 Å Release Date: 2025-12-24 Classification: OXIDOREDUCTASE Ligands: SF4, A1IW2, CL, LI |
Organism: Desulfovibrio desulfuricans
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: SF4, A1IW2, CL, LI
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Crystal Structure Of Small Molecule Ars-1620 Covalently Bound To K-Ras G12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2018-02-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, 91S, GOL, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: CA, 91S, GOL, GDP
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-Ethyl-7-[(3-Methoxypropyl)Amino] -3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.0,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50Y
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-7-[(Dimethyl-1,3-Thiazol-2-Yl)Amino]-10-Ethyl-3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.02,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50W
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-[(2S)-2,3-Dihydroxypropyl]-3-Methyl-7-(Methylamino)-3,5,8,10-Tetraazatricyclo [7.3.0.02,6]Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50O
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Crystal Structure Of Janus Kinase 2 In Complex With N,N-Dicyclopropyl-10-Ethyl-7-[(3-Methoxypropyl)Amino] -3-Methyl-3,5,8,10-Tetraazatricyclo[7.3.0.0,6] Dodeca-1(9),2(6),4,7,11-Pentaene-11-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-08-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 50V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-26
Ligands: 50V
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Crystal Structure Of Janus Kinase 2 In Complex With A 9H-Carbazole-1-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-06-03 Classification: Transferase/Transferase Inhibitor Ligands: 4OK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4OK
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Structure Of Janus Kinase 2 With A Pyrrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-02-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-16
Ligands: J2I
