Search Count: 8
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Dyrk1A Kinase Domain In Complex With A 6-Azaindole Derivative, Gnf2133.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2020-03-04 Classification: TRANSFERASE Ligands: Q8J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: Q8J
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Trastuzumab Fab D185A (Light Chain) Mutant.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-02-14 Classification: IMMUNE SYSTEM Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-14
Ligands: EDO
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Trastuzumab Fab N158A, D185A, K190A (Light Chain) Triple Mutant.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2018-02-14 Classification: IMMUNE SYSTEM Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-14
Ligands: EDO
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Trastuzumab Fab D185A (Light Chain) Mutant Biotin Conjugation.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-02-14 Classification: IMMUNE SYSTEM Ligands: EDO, BTN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-14
Ligands: EDO, BTN
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-06-03 Classification: Transferase/Transferase inhibitor Ligands: 4EJ, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4EJ, GOL, CL
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2015-06-03 Classification: Transferase/Transferase inhibitor Ligands: 4EK, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4EK, SO4, GOL
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(R)-2-Phenylpyrrolidine Substitute Imidazopyridazines: A New Class Of Potent And Selective Pan-Trk Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-06-03 Classification: Transfease/Transferase Inhibitor Ligands: 4F6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-03
Ligands: 4F6, SO4
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Discovery Of A Selective Trk Inhibitor With Efficacy In Rodent Cancer Tumor Models
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, 0F4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: CL, 0F4
