Search Count: 15
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Crystal Structure Of Ap2 Associated Kinase 1 Complexed With 5-[(4-Aminopiperidin-1-Yl)Methyl]-N-{3-[5-(Propan-2-Yl)-1,3,4-Thiadiazol-2-Yl]Phenyl}Pyrrolo[2,1-F][1,2,4]Triazin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-07-12 Classification: TRANSFERASE Ligands: YFV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: YFV, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Complexed With (5P)-3-({(8R)-5-[(4-Aminopiperidin-1-Yl)Methyl]Pyrrolo[2,1-F][1,2,4]Triazin-4-Yl}Amino)-5-[2-(Propan-2-Yl)-2H-Tetrazol-5-Yl]Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-07-12 Classification: TRANSFERASE Ligands: ZRR, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: ZRR, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YFV, SO4, 5OI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: YFV, SO4, 5OI
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand 2-(1-Amino-3-Methylbutyl)-6- (Pyridin-4-Yl)Quinoline-4-Carbonitrile
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5P6, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5P6, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5QI, PG6, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5QI, PG6, SO4, YFV
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand N-[3-Methoxy-4-(1,3-Oxazol-5-Yl)Phenyl]-3-(Propan-2-Yl)Piperidine-2-Carboxamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: YFS, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: YFS, SO4, YFV
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-Methoxy-4- (1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: YFY, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: YFY, SO4, YFV
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: Z3A
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 9J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 9J4
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Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2015-09-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4UQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4UQ
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Crystal Structure Of Bruton Agammaglobulinemia Tyrosine Kinase Complexed With Bms-824171 Aka 6-[(3R)-3-(4-Tert-Bu Tylbenzamido)Piperidin-1-Yl]-2-{[4-(Morpholine-4-Carbonyl) Phenyl]Amino}Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2015-09-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4US, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: 4US, DMS, EDO
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Structure Of A Carboxamide Compound (3) (2-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}-4-Oxo-4H-1Lambda~4~,3-Thiazole-5-Carboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WE
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Structure Of A Carvoxamide Compound (15) (N-[4-(Isoquinolin-7-Yl)Pyridin-2-Yl]Cyclopropanecarboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WF
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Structure Of A Carboxamine Compound (26) (2-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}-4-Methoxypyrimidine-5-Carboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WG
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE/INHIBITOR Ligands: 3QX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3QX