Search Count: 38
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Crystal Structure Of Casein Kinase 2 (Ck2) Alpha In Complex With Bms-595
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: A1DAS, MN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1DAS, MN, CL
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Crystal Structure Of Ap2 Associated Kinase 1 Complexed With 5-[(4-Aminopiperidin-1-Yl)Methyl]-N-{3-[5-(Propan-2-Yl)-1,3,4-Thiadiazol-2-Yl]Phenyl}Pyrrolo[2,1-F][1,2,4]Triazin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-07-12 Classification: TRANSFERASE Ligands: YFV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: YFV, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Complexed With (5P)-3-({(8R)-5-[(4-Aminopiperidin-1-Yl)Methyl]Pyrrolo[2,1-F][1,2,4]Triazin-4-Yl}Amino)-5-[2-(Propan-2-Yl)-2H-Tetrazol-5-Yl]Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-07-12 Classification: TRANSFERASE Ligands: ZRR, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: ZRR, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YFV, SO4, 5OI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: YFV, SO4, 5OI
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand 2-(1-Amino-3-Methylbutyl)-6- (Pyridin-4-Yl)Quinoline-4-Carbonitrile
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5P6, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5P6, SO4
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-(Difluorom Ethoxy)-4-(1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2022-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5QI, PG6, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: 5QI, PG6, SO4, YFV
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand N-[3-Methoxy-4-(1,3-Oxazol-5-Yl)Phenyl]-3-(Propan-2-Yl)Piperidine-2-Carboxamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: YFS, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: YFS, SO4, YFV
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Crystal Structure Of Ap2 Associated Kinase 1 Isoform 1 Complexed With Ligand (2R)-2-Amino-N-[3-Methoxy-4- (1,3-Oxazol-5-Yl)Phenyl]-4-Methylpentanamide
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-28 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: YFY, SO4, YFV |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: YFY, SO4, YFV
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With 6-[1-(2,2-Difluoroethyl)-4-(6-Methylpyridin-2-Yl)-1H-Imidazol-5-Yl]Imidazo[1,2-A]Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2020-02-05 Classification: TRANSFERASE Ligands: QMY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: QMY, GOL
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With 6-[4-(3-Chloro-4-Fluorophenyl)-1-(2-Hydroxyethyl)-1H-Imidazol-5-Yl]Imidazo[1,2-B]Pyridazine-3-Carbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2020-02-05 Classification: TRANSFERASE Ligands: QMV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: QMV, GOL
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: Z3A
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(6-Fluoropyridin-3-Yl)-4-Oxo-4,5,6,7-Tetrahydro-1H-Pyrrolo[3,2-C]Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2M, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2M, GOL
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(6-Methoxypyridin-3-Yl)-1H-Pyrrolo[3,2-B]Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2V
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(5-Methoxypyridin-2-Yl)-1H-Pyrrolo[3,2-B] Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2Y, GOL
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Tgf-Beta Receptor Type 2 Kinase Domain In Complex With N- {4-[3-(6-Methoxypyridin-3-Yl)-1H-Pyrrolo[3,2-B]Pyridin-2- Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2V, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2V, MG, GOL
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-(3-Fluoropyridin-4-Yl)-2-[6-(Trifluoromethyl)Pyridin-2-Yl]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-02-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: D0A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: D0A
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Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 9J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 9J4
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Crystal Structure Of Gsk3B In Complex With Compound 15: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Methoxypyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UO
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Crystal Structure Of Gsk3B In Complex With Compound 18: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Phenylpyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UP