Search Count: 29
![]() |
Structure Of Akt1(E17K) With Compound 3
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2024-09-04 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOO, SO4, ZN |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: EDO, XOO, SO4, ZN
![]() |
Structure Of Akt1(E17K) With Compound 3 (Zinc-Free)
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2024-09-04 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOO, SO4 |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: EDO, XOO, SO4
![]() |
Structure Of Akt1(Wt) With Compound 3
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2024-09-04 Classification: TRANSFERASE/INHIBITOR Ligands: EDO, XOO, SO4 |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: EDO, XOO, SO4
![]() |
Structure Of Akt1(E17K) With Compound 4
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-09-04 Classification: TRANSFERASE/INHIBITOR Ligands: XQ2, EDO, SO4, ZN, CL |
Organism: Homo sapiens, Lama glama
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: XQ2, EDO, SO4, ZN, CL
![]() |
Structure Of Akt2 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2024-09-04 Classification: TRANSFERASE/INHIBITOR Ligands: XOO, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: XOO, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-11-06 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: MG, GDP, MOV
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O67 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O67
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5V
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, O5Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: MG, GDP, O5Y
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To An Acryloylazetidine Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Inhibitor Ligands: CA, GDP, O5S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: CA, GDP, O5S
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With An Imidazopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-09 Classification: transferase/transferase inhibitor Ligands: 6YN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6YN
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL
![]() |
Co-Crystal Structure Of Pim1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3UR
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With An Aminooxadiazole-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 38W, GOL
