Search Count: 25
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The Crystal Structure Of A Mouse Fab Fragment Tl1 In Complex With A Human Glucose-6-Phosphate Isomerase Peptide 293-307
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2022-12-21 Classification: IMMUNE SYSTEM |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2022-12-21
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Human P300 Complexed With A Proline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C0C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C0C
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Human P300 Complexed With A Glycine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EDO, C3I, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ZN, EDO, C3I, ACT
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Human P300 Complexed With An Azaindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: TRANSFERASE/INHIBITOR Ligands: ETL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: ETL
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Alpha-1 Antitrypsin C232S Complexed With Cmpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-04-07 Classification: UNKNOWN FUNCTION Ligands: GOL, UL2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: GOL, UL2
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Alpha-1 Antitrypsin (C232S) Complexed With Cmpd 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2021-04-07 Classification: UNKNOWN FUNCTION Ligands: UKZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: UKZ, GOL
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Alpha 1-Antitrypsin (C232S) Complexed With Gsk716
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-03-10 Classification: PROTEIN BINDING Ligands: R7Z, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: R7Z, SO4
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Pi3K Alpha Lipid Kinase With Active Site Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-06-17 Classification: Transferase/Transferase Inhibitor Ligands: 4EL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 4EL
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk147
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3YZ
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk199
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3Z0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3Z0
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 11C [N-{2-[1-(6-Carbamoylthieno[3,2-D]Pyrimidin-4-Yl)Piperidin-4-Yl]Ethyl}-N'-Ethylthiophene-2,5-Dicarboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NQ
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 28 [4-(4-{2-[(2,2-Dimethylpropanoyl)Amino]Ethyl}Piperidin-1-Yl)Thieno[3,2-D]Pyrimidine-6-Carboxamide[
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NR
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 3 [14-(4-{2-[(Methylsulfonyl)Amino]Ethyl}Piperidin-1-Yl)Thieno[3,2-D]Pyrimidine-6-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NS, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NS, GOL, NA
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Crystal Structure Of An Extender (Spd28345)-Modified Human Pdk1 Complex 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: SYP
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Pdk1 In Complex With Dfg-Out Inhibitor Xxx
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-04-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MP7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: MP7
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Crystal Structure Of Aurora A In Complex With Tpx2 And Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2009-08-04 Classification: TRANSFERASE Ligands: 2JZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-08-04
Ligands: 2JZ
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The Complex Structure Of The Map Kinase P38/Compound 14B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2009-08-04 Classification: TRANSFERASE Ligands: 5JZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-08-04
Ligands: 5JZ
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-(1-Benzyl-Piperidin-4-Yl)-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1H
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With N-[1-(2,6-Dimethoxy-Benzyl)-Piperidin-4-Yl]-4-Mercapto-Butyramide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1I
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Crystal Structure Of The Human Bace1 Catalytic Domain In Complex With 4-(4-Fluoro-Benzyl)-Piperazine-2-Carboxylic Acid (2-Mercapto-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-01-20 Classification: HYDROLASE Ligands: F1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-20
Ligands: F1J
