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7APQ image
The Fk1 Domain Of Fkbp51 In Complex With (1S,5S,6R)-10-(Benzo[D]Thiazol-6-Ylsulfonyl)-5-(Methoxymethyl)-3-(Pyridin-2-Ylmethyl)-3,10-Diazabicyclo[4.3.1]Decan-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.09 Å Release Date: 2021-11-10
Classification: ISOMERASE
Ligands: RQW

7APT image
The Fk1 Domain Of Fkbp51 In Complex With ((1S,5S,6R)-10-((3,5-Dichlorophenyl)Sulfonyl)-2-Oxo-5-Vinyl-3,10-Diazabicyclo[4.3.1]Decan-3-Yl)Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.13 Å Release Date: 2021-11-10
Classification: ISOMERASE
Ligands: RRZ

7APW image
The Fk1 Domain Of Fkbp51 In Complex With (1S,5S,6R)-10-(Benzo[D]Thiazol-6-Ylsulfonyl)-5-(Methoxymethyl)-3-(Pyridin-2-Ylethyl)-3,10-Diazabicyclo[4.3.1]Decan-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.89 Å Release Date: 2021-11-10
Classification: CHAPERONE
Ligands: RSB

7APS image
The Fk1 Domain Of Fkbp51 In Complex With (2S)-2-((1S,5R,6R)-10-((3,5-Dichlorophenyl)Sulfonyl)-2-Oxo-5-Vinyl-3,10-Diazabicyclo[4.3.1]Decan-3-Yl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:0.94 Å Release Date: 2021-11-03
Classification: ISOMERASE
Ligands: RR5

6JZ0 image
Crystal Structure Of Egfr Kinase Domain In Complex With Compound 78
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.86 Å Release Date: 2019-12-04
Classification: TRANSFERASE/INHIBITOR
Ligands: CKO

3M11 image
Crystal Structure Of Aurora A Kinase Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.75 Å Release Date: 2011-03-09
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: AKI

3GBK image
Crystal Structure Of Human Ppar-Gamma Ligand Binding Domain Complexed With A Potent And Selective Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2009-12-29
Classification: ligand binding protein
Ligands: 2PQ

2X0I image
2.9 A Resolution Structure Of Malate Dehydrogenase From Archaeoglobus Fulgidus In Complex With Nadh
Organism: Archaeoglobus fulgidus dsm 4304
Method: X-RAY DIFFRACTION
Resolution:2.91 Å Release Date: 2009-12-22
Classification: OXIDOREDUCTASE
Ligands: NAI, SO4, NA

2X0J image
2.8 A Resolution Structure Of Malate Dehydrogenase From Archaeoglobus Fulgidus In Complex With Etheno-Nad
Organism: Archaeoglobus fulgidus dsm 4304
Method: X-RAY DIFFRACTION
Resolution:2.79 Å Release Date: 2009-12-22
Classification: OXIDOREDUCTASE
Ligands: ENA, SO4

3FDN image
Structure-Based Drug Design Of Novel Aurora Kinase A Inhibitors: Structure Basis For Potency And Specificity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2009-09-15
Classification: TRANSFERASE
Ligands: MMH

2HWQ image
Structural Basis For The Structure-Activity Relationships Of Peroxisome Proliferator-Activated Receptor Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2007-08-07
Classification: LIGAND BINDING PROTEIN
Ligands: DRY

2HWR image
Structural Basis For The Structure-Activity Relationships Of Peroxisome Proliferator-Activated Receptor Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.34 Å Release Date: 2007-08-07
Classification: LIGAND BINDING PROTEIN
Ligands: DRD

2ATH image
Crystal Structure Of The Ligand Binding Domain Of Human Ppar-Gamma Im Complex With An Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.28 Å Release Date: 2006-08-25
Classification: TRANSCRIPTION
Ligands: 3EA

2G0G image
Structure-Based Drug Design Of A Novel Family Of Ppar Partial Agonists: Virtual Screening, X-Ray Crystallography And In Vitro/In Vivo Biological Activities
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.54 Å Release Date: 2006-05-16
Classification: TRANSCRIPTION ACTIVATOR
Ligands: SP0

2G0H image
Structure-Based Drug Design Of A Novel Family Of Ppar Partial Agonists: Virtual Screening, X-Ray Crystallography And In Vitro/In Vivo Biological Activities
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2006-05-16
Classification: TRANSCRIPTION ACTIVATOR
Ligands: SP3

2F4B image
Crystal Structure Of The Ligand Binding Domain Of Human Ppar-Gamma In Complex With An Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.07 Å Release Date: 2006-02-14
Classification: TRANSCRIPTION ACTIVATOR
Ligands: EHA
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