Search Count: 15
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX7, IOD, 1HX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX7, IOD, 1HX
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Crystal Structure Of An Allosteric Inhibitor Bound To Human Ripk1 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2025-12-24 Classification: IMMUNE SYSTEM Ligands: A1IX9, IOD, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IX9, IOD, PEG
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Crystal Structure Of The Indoleamine 2,3-Dioxygenase 1 (Ido1) In Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2021-09-29 Classification: IMMUNOSUPPRESSANT Ligands: SLW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-29
Ligands: SLW
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Crystal Structure Of The Indoleamine 2,3-Dioxygenagse 1 (Ido1) Complexed With Iacs-70099
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2021-09-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: YRP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-01
Ligands: YRP
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Crystal Structure Of The Indoleamine 2,3-Dioxygenagse 1 (Ido1) Complexed With Iacs-8968
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-09-01 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: YRM, HEM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-01
Ligands: YRM, HEM
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B-Raf Wild-Type Kinase Domain In Complex With A Purinylpyridinylamino-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2016-05-04 Classification: Transferase/Transferase Inhibitor Ligands: 5XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5XJ
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Crystal Structure Of Pi3K-Gamma In Complex With Imidazopyridazine 19E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2013-04-10 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 0U0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-10
Ligands: SO4, 0U0
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Crystal Structure Of Pi3K-Gamma In Complex With Imidazopyridine 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-07-18 Classification: Transferase/Inhibitor Ligands: SO4, 0TZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-18
Ligands: SO4, 0TZ
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Crystal Structure Of Human Anaplastic Lymphoma Kinase In Complex With Acyliminobenzimidazole Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-07-11 Classification: Transferase/Inhibitor Ligands: 0US |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0US
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Crystal Structure Of Human Anaplastic Lymphoma Kinase In Complex With Acyliminobenzimidazole Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2012-07-11 Classification: Transferase/Inhibitor Ligands: 0UU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0UU
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Crystal Structure Of Human Anaplastic Lymphoma Kinase In Complex With Acyliminobenzimidazole Inhibitor 36
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-07-11 Classification: Transferase/Inhibitor Ligands: 0UV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0UV, GOL
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Crystal Structure Of C-Met In Complex With Triazolopyridazine Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0JJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0JJ
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Crystal Structure Of C-Met In Complex With Triazolopyridinone Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0JK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0JK
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Crystal Structure Of C-Met In Complex With Triazolopyridinone Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-05-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0JL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-30
Ligands: 0JL
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Crystal Structure Of Human Anaplastic Lymphoma Kinase In Complex With A Piperidine-Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2012-02-08 Classification: Transferase/Inhibitor Ligands: 0JF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: 0JF
