Search Count: 14
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Crystal Structure Of Human Clk1 Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
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Crystal Structure Of Human Acvr1 (Alk2) Kinase In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2024-11-06 Classification: SIGNALING PROTEIN Ligands: SO4, XQX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: SO4, XQX
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Crystal Structure Of Fgfr4 With An Irreversible Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2015-04-01 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 40M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-01
Ligands: SO4, 40M
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Discovery And Optimization Of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-15 Classification: TRANSFERASE Ligands: J82 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: J82
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Crystal Structure Of Apo Human Prpf4B Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2013-08-28 Classification: TRANSFERASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: SO4
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Crystal Structure Of Adp-Bound Human Prpf4B Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2013-08-28 Classification: TRANSFERASE Ligands: ADP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: ADP, SO4
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Crystal Structure Of Amppnp-Bound Human Prpf4B Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-08-28 Classification: TRANSFERASE Ligands: ANP, SO4, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: ANP, SO4, MG
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Crystal Structure Of Human Prpf4B Kinase Domain In Complex With 4-{5-[(2-Chloro-Pyridin-4-Ylmethyl)-Carbamoyl]-Thiophen-2-Yl}-Benzo[B]Thiophene-2-Carboxylic Acid Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2013-08-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1EH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: 1EH, SO4
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X-Ray Structure Of Pi3K-Gamma Bound To A 4-(Morpholin-4-Yl)- (6-Oxo-1,6-Dihydropyrimidin-2-Yl)Amide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2012-11-14 Classification: Transferase/Transferase Inhibitor Ligands: 0W7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0W7
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Discovery And Optimization Of New Benzimidazole- And Benzoxazole-Pyrimidone Selective Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-05-16 Classification: TRANSFERASE Ligands: VWN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: VWN
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Crystal Structure Of Cdk4 In Complex With A D-Type Cyclin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2009-03-10 Classification: CELL CYCLE Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: GOL
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Crystal Structure Of Cdk4 In Complex With A D-Type Cyclin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2009-03-10 Classification: CELL CYCLE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
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Crystal Structure Of Cdk4 In Complex With A D-Type Cyclin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2009-03-10 Classification: CELL CYCLE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
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Crystal Structure Of Cdk4 In Complex With A D-Type Cyclin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2009-03-10 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
