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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 2-Amino-N-(5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-04-22 Classification: TRANSFERASE Ligands: A1ER0 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor 4-((5-((5-Chloro-4-(((3R,3Ar,6R,6Ar)-6-Methoxyhexahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-((2-(Dimethylamino)Ethyl)(Methyl)Amino)Phenyl)Carbamoyl)-1-Methyl-3H-Pyrazol-1-Ium-3-Ide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ER9 |
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Crystal Structure Of The Nuak1-Mark3 Kinase Domain Chimera Bound With Small Molecule Inhibitor N-(5-((5-Chloro-4-(((3As,6R,6Ar)-6-Methoxy-3A,5,6,6A-Tetrahydrofuro[3,2-B]Furan-3-Yl)Oxy)Pyrimidin-2-Yl)Amino)-2-(((2R,7Ar)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl)Methoxy)Phenyl)-1-Methyl-1H-Pyrazole-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2026-04-22 Classification: CYTOSOLIC PROTEIN Ligands: A1ESF |
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Site-Specific Introduction Of Sulfoxides And Sulfones Into Polyketide Scaffold Through A Relayed Chemo-Biosynthetic Strategy
Organism: Streptomyces armeniacus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2025-01-22 Classification: BIOSYNTHETIC PROTEIN |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-11-22 Classification: GENE REGULATION/DNA Ligands: ZN, SAM |
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Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-11-15 Classification: GENE REGULATION/DNA Ligands: ZN, SAM |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2022-04-20 Classification: TRANSFERASE Ligands: JAU |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-07-21 Classification: TRANSCRIPTION Ligands: EDO, ZN |
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Organism: Amycolatopsis mediterranei (strain u-32)
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-07-04 Classification: OXIDOREDUCTASE Ligands: HEM |
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Organism: Amycolatopsis mediterranei (strain u-32)
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-07-04 Classification: OXIDOREDUCTASE Ligands: HEM, 9LF |
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Crystal Structure Analysis Of The Superoxide Dismutase From Clostridium Difficile
Organism: Clostridium difficile
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-08-29 Classification: OXIDOREDUCTASE Ligands: FE |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2007-07-31 Classification: TRANSPORT PROTEIN |












