Search Count: 15
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Discovery Of A Small Molecule Itk And Pan-Trk Kinase Inhibitor (Pf-07245303) For The Potential Topical Treatment Of Atopic Dermatitis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-11-19 Classification: SIGNALING PROTEIN Ligands: A1B66 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-19
Ligands: A1B66
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Pad2 With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-07-30 Classification: HYDROLASE Ligands: A1CE0, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1CE0, CA
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-05-28 Classification: HYDROLASE Ligands: CA, A1A8O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1A8O
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Inhibiting Peptidylarginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, A1BZK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: CA, A1BZK
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Potent Inhibition Of The Protein Arginine Deiminases (Pad1-4) By Targeting A Ca2+ Dependent Allosteric Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2025-05-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: A1A9P, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-28
Ligands: A1A9P, 3YZ
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Crystal Structure Of Irak4 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2024-05-01 Classification: TRANSFERASE Ligands: A1AFO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-01
Ligands: A1AFO
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Crystal Structure Of Irak4 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2024-05-01 Classification: TRANSFERASE Ligands: A1AFH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-01
Ligands: A1AFH
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 5 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: LKY, 4Y5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: LKY, 4Y5, SO4
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 6A Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XNR, 4Y5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XNR, 4Y5
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Human Retenoid-Related Orphan Receptor-Gamma (Rorc2) Ligand-Binding Domain In Complex With Compound 8 Andindazole Acid Bound In H12-Pocket
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-03-01 Classification: DNA BINDING PROTEIN Ligands: XO5, XNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-01
Ligands: XO5, XNX
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Crystal Structure Of Irak4 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BV
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Crystal Structure Of Irak4 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8BY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8BY
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Crystal Structure Of Irak4 In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8C1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8C1
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Crystal Structure Of Irak4 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8CD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8CD
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Crystal Structure Of Irak4 In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2017-05-24 Classification: TRANSFERASE Ligands: 8CG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 8CG